Overkleeft HS - Search Results

1

Structure-based design of β1i or β5i specific inhibitors of human immunoproteasomes.

de Bruin G, Huber EM, Xin BT, van Rooden EJ, Al-Ayed K, Kim KB, Kisselev AF, Driessen C, van der Stelt M, van der Marel GA, Groll M, Overkleeft HS. de Bruin G, et al. Among authors: overkleeft hs. J Med Chem. 2014 Jul 24;57(14):6197-209. doi: 10.1021/jm500716s. Epub 2014 Jul 15. J Med Chem. 2014. PMID: 25006746

2

Extended peptide-based inhibitors efficiently target the proteasome and reveal overlapping specificities of the catalytic beta-subunits.

Kessler BM, Tortorella D, Altun M, Kisselev AF, Fiebiger E, Hekking BG, Ploegh HL, Overkleeft HS. Kessler BM, et al. Among authors: overkleeft hs. Chem Biol. 2001 Sep;8(9):913-29. doi: 10.1016/s1074-5521(01)00069-2. Chem Biol. 2001. PMID: 11564559

3

Solid-phase synthesis of cyclic RGD-furanoid sugar amino acid peptides as integrin inhibitors.

van Well RM, Overkleeft HS, van der Marel GA, Bruss D, Thibault G, de Groot PG, van Boom JH, Overhand M. van Well RM, et al. Among authors: overkleeft hs. Bioorg Med Chem Lett. 2003 Feb 10;13(3):331-4. doi: 10.1016/s0960-894x(02)01022-3. Bioorg Med Chem Lett. 2003. PMID: 12565923

4

Synthesis and biological evaluation of novel turn-modified gramicidin S analogues.

Grotenbreg GM, Spalburg E, de Neeling AJ, van der Marel GA, Overkleeft HS, van Boom JH, Overhand M. Grotenbreg GM, et al. Among authors: overkleeft hs. Bioorg Med Chem. 2003 Jul 3;11(13):2835-41. doi: 10.1016/s0968-0896(03)00219-0. Bioorg Med Chem. 2003. PMID: 12788356

5

The caspase-like sites of proteasomes, their substrate specificity, new inhibitors and substrates, and allosteric interactions with the trypsin-like sites.

Kisselev AF, Garcia-Calvo M, Overkleeft HS, Peterson E, Pennington MW, Ploegh HL, Thornberry NA, Goldberg AL. Kisselev AF, et al. Among authors: overkleeft hs. J Biol Chem. 2003 Sep 19;278(38):35869-77. doi: 10.1074/jbc.M303725200. Epub 2003 Jun 18. J Biol Chem. 2003. PMID: 12815064 Free article.

6

Chemistry in living cells: detection of active proteasomes by a two-step labeling strategy.

Ovaa H, van Swieten PF, Kessler BM, Leeuwenburgh MA, Fiebiger E, van den Nieuwendijk AM, Galardy PJ, van der Marel GA, Ploegh HL, Overkleeft HS. Ovaa H, et al. Among authors: overkleeft hs. Angew Chem Int Ed Engl. 2003 Aug 11;42(31):3626-9. doi: 10.1002/anie.200351314. Angew Chem Int Ed Engl. 2003. PMID: 12916032 No abstract available.

7

The use of a mannitol-derived fused oxacycle as a combinatorial scaffold.

Timmer MS, Verdoes M, Sliedregt LA, van der Marel GA, van Boom JH, Overkleeft HS. Timmer MS, et al. Among authors: overkleeft hs. J Org Chem. 2003 Nov 28;68(24):9406-11. doi: 10.1021/jo0349429. J Org Chem. 2003. PMID: 14629165

8

Olefin metathesis in glycobiology: new routes towards diverse neoglycoconjugates.

Leeuwenburgh MA, van der Marel GA, Overkleeft HS. Leeuwenburgh MA, et al. Among authors: overkleeft hs. Curr Opin Chem Biol. 2003 Dec;7(6):757-65. doi: 10.1016/j.cbpa.2003.10.009. Curr Opin Chem Biol. 2003. PMID: 14644186 Review.

9

A short route toward chiral, polyhydroxylated indolizidines and quinolizidines.

Verhelst SH, Paez Martinez B, Timmer MS, Lodder G, van der Marel GA, Overkleeft HS, van Boom JH. Verhelst SH, et al. Among authors: overkleeft hs. J Org Chem. 2003 Dec 12;68(25):9598-603. doi: 10.1021/jo0350662. J Org Chem. 2003. PMID: 14656083

10

A novel strategy towards the synthesis of orthogonally functionalised 4-aminoglycosides.

van den Bos LJ, Codée JD, van Boom JH, Overkleeft HS, van der Marel GA. van den Bos LJ, et al. Among authors: overkleeft hs. Org Biomol Chem. 2003 Dec 7;1(23):4160-5. doi: 10.1039/b309823k. Epub 2003 Oct 21. Org Biomol Chem. 2003. PMID: 14685319

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