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Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
---|---|
2008 | 2 |
2009 | 3 |
2024 | 0 |
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4 results
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Page 1
Exploiting structural analysis, in silico screening, and serendipity to identify novel inhibitors of drug-resistant falciparum malaria.
ACS Chem Biol. 2009 Jan 16;4(1):29-40. doi: 10.1021/cb8002804.
ACS Chem Biol. 2009.
PMID: 19146480
Free PMC article.
Novel non-active site inhibitor of Cryptosporidium hominis TS-DHFR identified by a virtual screen.
Martucci WE, Udier-Blagovic M, Atreya C, Babatunde O, Vargo MA, Jorgensen WL, Anderson KS.
Martucci WE, et al.
Bioorg Med Chem Lett. 2009 Jan 15;19(2):418-23. doi: 10.1016/j.bmcl.2008.11.054. Epub 2008 Nov 20.
Bioorg Med Chem Lett. 2009.
PMID: 19059777
Free PMC article.
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Disruption of the crossover helix impairs dihydrofolate reductase activity in the bifunctional enzyme TS-DHFR from Cryptosporidium hominis.
Vargo MA, Martucci WE, Anderson KS.
Vargo MA, et al.
Biochem J. 2009 Feb 1;417(3):757-64. doi: 10.1042/BJ20081247.
Biochem J. 2009.
PMID: 18851711
Free PMC article.
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Explaining an unusually fast parasitic enzyme: folate tail-binding residues dictate substrate positioning and catalysis in Cryptosporidium hominis thymidylate synthase.
Martucci WE, Vargo MA, Anderson KS.
Martucci WE, et al.
Biochemistry. 2008 Aug 26;47(34):8902-11. doi: 10.1021/bi800466z. Epub 2008 Aug 2.
Biochemistry. 2008.
PMID: 18672899
Free PMC article.
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