Rastelli G - Search Results

1

Insights into the interaction of negative allosteric modulators with the metabotropic glutamate receptor 5: discovery and computational modeling of a new series of ligands with nanomolar affinity.

Anighoro A, Graziani D, Bettinelli I, Cilia A, De Toma C, Longhi M, Mangiarotti F, Menegon S, Pirona L, Poggesi E, Riva C, Rastelli G. Anighoro A, et al. Among authors: rastelli g. Bioorg Med Chem. 2015 Jul 1;23(13):3040-58. doi: 10.1016/j.bmc.2015.05.008. Epub 2015 May 12. Bioorg Med Chem. 2015. PMID: 26014480

2

Conformational analysis of phthalein derivatives acting as thymidylate synthase inhibitors by means of 1H NMR and quantum chemical calculations.

Ghelli S, Rastelli G, Barlocco D, Rinaldi M, Tondi D, Pecorari P, Costi MP. Ghelli S, et al. Among authors: rastelli g. Bioorg Med Chem. 1996 Oct;4(10):1783-94. doi: 10.1016/0968-0896(96)00193-9. Bioorg Med Chem. 1996. PMID: 8931948

3

Molecular dynamics simulations of the structure of aldose reductase complexed with the inhibitor tolrestat.

Rastelli G, Costantino L. Rastelli G, et al. Bioorg Med Chem Lett. 1998 Mar 17;8(6):641-6. doi: 10.1016/s0960-894x(98)00083-3. Bioorg Med Chem Lett. 1998. PMID: 9871575

4

1-Benzopyran-4-one antioxidants as aldose reductase inhibitors.

Costantino L, Rastelli G, Gamberini MC, Vinson JA, Bose P, Iannone A, Staffieri M, Antolini L, Del Corso A, Mura U, Albasini A. Costantino L, et al. Among authors: rastelli g. J Med Chem. 1999 Jun 3;42(11):1881-93. doi: 10.1021/jm980441h. J Med Chem. 1999. PMID: 10354396

5

Isoxazolo-[3,4-d]-pyridazin-7-(6H)-one as a potential substrate for new aldose reductase inhibitors.

Costantino L, Rastelli G, Gamberini MC, Giovannoni MP, Dal Piaz V, Vianello P, Barlocco D. Costantino L, et al. Among authors: rastelli g. J Med Chem. 1999 Jun 3;42(11):1894-900. doi: 10.1021/jm981107o. J Med Chem. 1999. PMID: 10354397

6

Interaction of pyrimethamine, cycloguanil, WR99210 and their analogues with Plasmodium falciparum dihydrofolate reductase: structural basis of antifolate resistance.

Rastelli G, Sirawaraporn W, Sompornpisut P, Vilaivan T, Kamchonwongpaisan S, Quarrell R, Lowe G, Thebtaranonth Y, Yuthavong Y. Rastelli G, et al. Bioorg Med Chem. 2000 May;8(5):1117-28. doi: 10.1016/s0968-0896(00)00022-5. Bioorg Med Chem. 2000. PMID: 10882022

7

Structural bases for the inhibition of aldose reductase by phenolic compounds.

Rastelli G, Antolini L, Benvenuti S, Costantino L. Rastelli G, et al. Bioorg Med Chem. 2000 May;8(5):1151-8. doi: 10.1016/s0968-0896(00)00052-3. Bioorg Med Chem. 2000. PMID: 10882025

8

Binding of 1-benzopyran-4-one derivatives to aldose reductase: a free energy perturbation study.

Rastelli G, Costantino L, Gamberini MC, Del Corso A, Mura U, Petrash JM, Ferrari AM, Pacchioni S. Rastelli G, et al. Bioorg Med Chem. 2002 May;10(5):1427-36. doi: 10.1016/s0968-0896(01)00408-4. Bioorg Med Chem. 2002. PMID: 11886805

9

Discovery of new inhibitors of aldose reductase from molecular docking and database screening.

Rastelli G, Ferrari AM, Costantino L, Gamberini MC. Rastelli G, et al. Bioorg Med Chem. 2002 May;10(5):1437-50. doi: 10.1016/s0968-0896(01)00410-2. Bioorg Med Chem. 2002. PMID: 11886806

10

Nitrophenyl derivatives as aldose reductase inhibitors.

Costantino L, Ferrari AM, Gamberini MC, Rastelli G. Costantino L, et al. Among authors: rastelli g. Bioorg Med Chem. 2002 Dec;10(12):3923-31. doi: 10.1016/s0968-0896(02)00318-8. Bioorg Med Chem. 2002. PMID: 12413844

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