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A Discovery Strategy for Selective Inhibitors of c-Src in Complex with the Focal Adhesion Kinase SH3/SH2-binding Region.
Chem Biol Drug Des. 2015 Aug;86(2):144-55. doi: 10.1111/cbdd.12473. Epub 2014 Nov 28.
Chem Biol Drug Des. 2015.
PMID: 25376742
Free PMC article.
Kinase consensus sequences: a breeding ground for crosstalk.
Rust HL, Thompson PR.
Rust HL, et al.
ACS Chem Biol. 2011 Sep 16;6(9):881-92. doi: 10.1021/cb200171d. Epub 2011 Jul 15.
ACS Chem Biol. 2011.
PMID: 21721511
Free PMC article.
Review.
Item in Clipboard
Using unnatural amino acid mutagenesis to probe the regulation of PRMT1.
Rust HL, Subramanian V, West GM, Young DD, Schultz PG, Thompson PR.
Rust HL, et al.
ACS Chem Biol. 2014 Mar 21;9(3):649-55. doi: 10.1021/cb400859z. Epub 2014 Jan 6.
ACS Chem Biol. 2014.
PMID: 24358983
Free PMC article.
Item in Clipboard
A combinatorial approach to characterize the substrate specificity of protein arginine methyltransferase 1.
Bicker KL, Obianyo O, Rust HL, Thompson PR.
Bicker KL, et al. Among authors: rust hl.
Mol Biosyst. 2011 Jan;7(1):48-51. doi: 10.1039/c0mb00015a. Epub 2010 Jul 6.
Mol Biosyst. 2011.
PMID: 20607165
Free PMC article.
Item in Clipboard
Mechanistic studies on transcriptional coactivator protein arginine methyltransferase 1.
Rust HL, Zurita-Lopez CI, Clarke S, Thompson PR.
Rust HL, et al.
Biochemistry. 2011 Apr 26;50(16):3332-45. doi: 10.1021/bi102022e. Epub 2011 Apr 1.
Biochemistry. 2011.
PMID: 21417440
Free PMC article.
Item in Clipboard
Automethylation of protein arginine methyltransferase 8 (PRMT8) regulates activity by impeding S-adenosylmethionine sensitivity.
Dillon MB, Rust HL, Thompson PR, Mowen KA.
Dillon MB, et al. Among authors: rust hl.
J Biol Chem. 2013 Sep 27;288(39):27872-80. doi: 10.1074/jbc.M113.491092. Epub 2013 Aug 14.
J Biol Chem. 2013.
PMID: 23946480
Free PMC article.
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