Weier RM - Search Results

1

Synthesis, crystal structure, and activity of pyrazole-based inhibitors of p38 kinase.

Graneto MJ, Kurumbail RG, Vazquez ML, Shieh HS, Pawlitz JL, Williams JM, Stallings WC, Geng L, Naraian AS, Koszyk FJ, Stealey MA, Xu XD, Weier RM, Hanson GJ, Mourey RJ, Compton RP, Mnich SJ, Anderson GD, Monahan JB, Devraj R. Graneto MJ, et al. Among authors: weier rm. J Med Chem. 2007 Nov 15;50(23):5712-9. doi: 10.1021/jm0611915. Epub 2007 Oct 19. J Med Chem. 2007. PMID: 17948975

2

Aminopyridinecarboxamide-based inhibitors: Structure-activity relationship.

Bonafoux DF, Bonar SL, Clare M, Donnelly AM, Glaenzer JL, Guzova JA, Huang H, Kishore NN, Koszyk FJ, Lennon PJ, Libby A, Mathialagan S, Oburn DS, Rouw SA, Sommers CD, Tripp CS, Vanella LJ, Weier R, Wolfson SG, Huang HC. Bonafoux DF, et al. Bioorg Med Chem. 2010 Jan 1;18(1):403-14. doi: 10.1016/j.bmc.2009.10.040. Epub 2009 Oct 27. Bioorg Med Chem. 2010. PMID: 19914076

3

1,2-Diarylimidazoles as potent, cyclooxygenase-2 selective, and orally active antiinflammatory agents.

Khanna IK, Weier RM, Yu Y, Xu XD, Koszyk FJ, Collins PW, Koboldt CM, Veenhuizen AW, Perkins WE, Casler JJ, Masferrer JL, Zhang YY, Gregory SA, Seibert K, Isakson PC. Khanna IK, et al. Among authors: weier rm. J Med Chem. 1997 May 23;40(11):1634-47. doi: 10.1021/jm9700225. J Med Chem. 1997. PMID: 9171873

4

Antiinflammatory 4,5-diarylimidazoles as selective cyclooxygenase inhibitors.

Barta TE, Stealey MA, Collins PW, Weier RM. Barta TE, et al. Among authors: weier rm. Bioorg Med Chem Lett. 1998 Dec 15;8(24):3443-8. doi: 10.1016/s0960-894x(98)00627-1. Bioorg Med Chem Lett. 1998. PMID: 9934449

5

Selective cyclooxygenase-2 inhibitors: heteroaryl modified 1,2-diarylimidazoles are potent, orally active antiinflammatory agents.

Khanna IK, Yu Y, Huff RM, Weier RM, Xu X, Koszyk FJ, Collins PW, Cogburn JN, Isakson PC, Koboldt CM, Masferrer JL, Perkins WE, Seibert K, Veenhuizen AW, Yuan J, Yang DC, Zhang YY. Khanna IK, et al. Among authors: weier rm. J Med Chem. 2000 Aug 10;43(16):3168-85. doi: 10.1021/jm0000719. J Med Chem. 2000. PMID: 10956225

6

A selective IKK-2 inhibitor blocks NF-kappa B-dependent gene expression in interleukin-1 beta-stimulated synovial fibroblasts.

Kishore N, Sommers C, Mathialagan S, Guzova J, Yao M, Hauser S, Huynh K, Bonar S, Mielke C, Albee L, Weier R, Graneto M, Hanau C, Perry T, Tripp CS. Kishore N, et al. J Biol Chem. 2003 Aug 29;278(35):32861-71. doi: 10.1074/jbc.M211439200. Epub 2003 Jun 17. J Biol Chem. 2003. PMID: 12813046 Free article.

7

1,2-Diarylpyrroles as potent and selective inhibitors of cyclooxygenase-2.

Khanna IK, Weier RM, Yu Y, Collins PW, Miyashiro JM, Koboldt CM, Veenhuizen AW, Currie JL, Seibert K, Isakson PC. Khanna IK, et al. Among authors: weier rm. J Med Chem. 1997 May 23;40(11):1619-33. doi: 10.1021/jm970036a. J Med Chem. 1997. PMID: 9171872

8

Inhibition of IKK-2 by 2-[(aminocarbonyl)amino]-5-acetylenyl-3-thiophenecarboxamides.

Bonafoux D, Bonar S, Christine L, Clare M, Donnelly A, Guzova J, Kishore N, Lennon P, Libby A, Mathialagan S, McGhee W, Rouw S, Sommers C, Tollefson M, Tripp C, Weier R, Wolfson S, Min Y. Bonafoux D, et al. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2870-5. doi: 10.1016/j.bmcl.2005.03.090. Bioorg Med Chem Lett. 2005. PMID: 15911271

9

Synthesis and antimineralocorticoid activities of some 6-substituted 7 alpha-carboalkoxy steroidal spirolactones.

Weier RM, Hofmann LM. Weier RM, et al. J Med Chem. 1977 Oct;20(10):1304-8. doi: 10.1021/jm00220a015. J Med Chem. 1977. PMID: 903917

10

Synthesis and gastrointestinal pharmacology of a 3E,5Z diene analogue of misoprostol.

Collins PW, Kramer SW, Gasiecki AF, Weier RM, Jones PH, Gullikson GW, Bianchi RG, Bauer RF. Collins PW, et al. Among authors: weier rm. J Med Chem. 1987 Jan;30(1):193-7. doi: 10.1021/jm00384a032. J Med Chem. 1987. PMID: 3100798

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