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Imidazo[1,2-a]quinoxalines for melanoma treatment with original mechanism of action.
Eur J Med Chem. 2021 Feb 15;212:113031. doi: 10.1016/j.ejmech.2020.113031. Epub 2020 Nov 24.
Eur J Med Chem. 2021.
PMID: 33309473
New imidazoquinoxaline derivatives: Synthesis, biological evaluation on melanoma, effect on tubulin polymerization and structure-activity relationships.
Zghaib Z, Guichou JF, Vappiani J, Bec N, Hadj-Kaddour K, Vincent LA, Paniagua-Gayraud S, Larroque C, Moarbess G, Cuq P, Kassab I, Deleuze-Masquéfa C, Diab-Assaf M, Bonnet PA.
Zghaib Z, et al.
Bioorg Med Chem. 2016 Jun 1;24(11):2433-2440. doi: 10.1016/j.bmc.2016.04.004. Epub 2016 Apr 1.
Bioorg Med Chem. 2016.
PMID: 27094151
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Imidazoquinoxaline anticancer derivatives and imiquimod interact with tubulin: Characterization of molecular microtubule inhibiting mechanisms in correlation with cytotoxicity.
Courbet A, Bec N, Constant C, Larroque C, Pugniere M, El Messaoudi S, Zghaib Z, Khier S, Deleuze-Masquefa C, Gattacceca F.
Courbet A, et al. Among authors: zghaib z.
PLoS One. 2017 Aug 10;12(8):e0182022. doi: 10.1371/journal.pone.0182022. eCollection 2017.
PLoS One. 2017.
PMID: 28797090
Free PMC article.
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Lipid nanocapsules formulation and cellular activities evaluation of a promising anticancer agent: EAPB0503.
Chouchou A, Aubert-Pouëssel A, Dorandeu C, Zghaib Z, Cuq P, Devoisselle JM, Bonnet PA, Bégu S, Deleuze-Masquefa C.
Chouchou A, et al. Among authors: zghaib z.
Int J Pharm Investig. 2017 Oct-Dec;7(4):155-163. doi: 10.4103/jphi.JPHI_53_17.
Int J Pharm Investig. 2017.
PMID: 29692974
Free PMC article.
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