A novel two-chain proteinase inhibitor generated by circularization of a multidomain precursor protein

Nat Struct Biol. 1999 Jun;6(6):526-30. doi: 10.1038/9293.

Abstract

Female reproductive tissues of the ornamental tobacco amass high levels of serine proteinase inhibitors (PIs) for protection against pests and pathogens. These PIs are produced from a precursor protein composed of six repeats each with a protease reactive site. Here we show that proteolytic processing of the precursor generates five single-chain PIs and a remarkable two-chain inhibitor formed by disulfide-bond linkage of N- and C-terminal peptide fragments. Surprisingly, PI precursors adopt this circular structure regardless of the number of inhibitor domains, suggesting this bracelet-like conformation is characteristic of the widespread potato inhibitor II (Pot II) protein family.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Binding Sites
  • Chymotrypsin / antagonists & inhibitors
  • Crystallization
  • Disulfides / chemistry
  • Disulfides / metabolism
  • Evolution, Molecular
  • Gene Duplication
  • Molecular Sequence Data
  • Molecular Weight
  • Nicotiana / chemistry
  • Nuclear Magnetic Resonance, Biomolecular
  • Peptide Fragments / chemistry*
  • Peptide Fragments / metabolism
  • Plant Proteins / chemistry*
  • Plant Proteins / isolation & purification
  • Plant Proteins / metabolism
  • Plant Structures / chemistry
  • Plants, Toxic
  • Protease Inhibitors*
  • Protein Conformation
  • Protein Folding
  • Protein Precursors / chemistry
  • Protein Precursors / metabolism*
  • Protein Structure, Secondary
  • Repetitive Sequences, Amino Acid
  • Serine Proteinase Inhibitors / chemistry*
  • Serine Proteinase Inhibitors / isolation & purification
  • Serine Proteinase Inhibitors / metabolism

Substances

  • Disulfides
  • Peptide Fragments
  • Plant Proteins
  • Protease Inhibitors
  • Protein Precursors
  • Serine Proteinase Inhibitors
  • proteinase inhibitor II protein, plant
  • proteinase inhibitor I (plants)
  • Chymotrypsin

Associated data

  • PDB/1QH2