Pentamidine is a potent inhibitor of [3H]idazoxan binding to imidazoline I2 receptors

Ann N Y Acad Sci. 1999 Jun 21:881:110-3. doi: 10.1111/j.1749-6632.1999.tb09349.x.
No abstract available

MeSH terms

  • Animals
  • Anti-Infective Agents / pharmacology
  • Binding Sites
  • Binding, Competitive
  • Cell Membrane / metabolism
  • Cryptosporidium / drug effects
  • Idazoxan / pharmacokinetics*
  • Imidazoline Receptors
  • Kinetics
  • Liver / metabolism
  • Pentamidine / analogs & derivatives*
  • Pentamidine / chemistry
  • Pentamidine / pharmacology*
  • Pneumocystis / drug effects
  • Radioligand Assay
  • Rats
  • Receptors, Drug / antagonists & inhibitors
  • Receptors, Drug / metabolism*

Substances

  • Anti-Infective Agents
  • Imidazoline Receptors
  • Receptors, Drug
  • Pentamidine
  • Idazoxan