Itch-scratch responses induced by opioids through central mu opioid receptors in mice

J Biomed Sci. 2000 May-Jun;7(3):248-52. doi: 10.1007/BF02255473.

Abstract

We examined scratch-inducing effects of intracisternal, intrathecal and intradermal injections of morphine and some opioid agonists in mice. Intracisternal injection of morphine (3 nmol/animal) and the mu-receptor agonist [D-Ala(2), N-Me-Phe(4), Gly(5)-ol]enkephalin (DAMGO; 0.2 nmol/animal) elicited scratching of the face, with little effect on scratching of the trunk. Intracisternal injection of the delta-receptor agonist [D-Pen(2,5)]enkephalin (DPDPE) and the kappa-receptor agonist U50488 were without effects. Intrathecal injection of morphine (0.1-3 nmol/animal) produced a dose-dependent increase in body scratching, with little effects on face scratching. Face scratching induced by intrathecal morphine (3 nmol/animal) was almost abolished by subcutaneous pretreatment with naloxone (1 mg/kg). Intradermal injections of morphine (3-100 nmol/site), DAMGO (1-100 nmol/site), DPDPE (10 and 100 nmol/site) and U50488 (10-100 nmol/site) did not elicit scratching of the site of injection. Intradermal injection of histamine (100 nmol/site) induced the scratching in ICR, but not ddY, mice and serotonin (30 and 50 nmol/site) elicited the scratching in either strain of mice. The results suggest that opioids induce scratching, and probably itching, through central mu-opioid receptors in the mouse.

MeSH terms

  • 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer / pharmacology
  • Analgesics, Opioid / pharmacology
  • Animals
  • Enkephalin, Ala(2)-MePhe(4)-Gly(5)- / pharmacology
  • Enkephalin, D-Penicillamine (2,5)- / pharmacology
  • Face / physiopathology
  • Histamine / pharmacology
  • Injections, Subcutaneous
  • Male
  • Mice
  • Mice, Inbred ICR
  • Mice, Inbred Strains
  • Morphine / pharmacology
  • Narcotics / agonists
  • Narcotics / pharmacology*
  • Pruritus / chemically induced*
  • Pruritus / physiopathology*
  • Receptors, Opioid, mu / physiology*
  • Serotonin / pharmacology
  • Sodium Chloride / administration & dosage
  • Sodium Chloride / pharmacology
  • Time Factors

Substances

  • Analgesics, Opioid
  • Narcotics
  • Receptors, Opioid, mu
  • Enkephalin, Ala(2)-MePhe(4)-Gly(5)-
  • Serotonin
  • Sodium Chloride
  • 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer
  • Morphine
  • Histamine
  • Enkephalin, D-Penicillamine (2,5)-