Comparison of the structure of vMIP-II with eotaxin-1, RANTES, and MCP-3 suggests a unique mechanism for CCR3 activation

Biochemistry. 2000 Oct 24;39(42):12837-44. doi: 10.1021/bi001166f.

Abstract

Herpesvirus-8 macrophage inflammatory protein-II (vMIP-II) binds a uniquely wide spectrum of chemokine receptors. We report the X-ray structure of vMIP-II determined to 2.1 A resolution. Like RANTES, vMIP-II crystallizes as a dimer and displays the conventional chemokine tertiary fold. We have compared the surface topology and electrostatic potential of vMIP-II to those of eotaxin-1, RANTES, and MCP-3, three CCR3 physiological agonists with known three-dimensional structures. Surface epitopes identified on RANTES to be involved in binding to CCR3 are mimicked on the eotaxin-1 and MCP-3 surface. However, the surface topology of vMIP-II in these regions is markedly different. The results presented here indicate that the structural basis for interaction with the chemokine receptor CCR3 by vMIP-II is different from that for the physiological agonists eotaxin-1, RANTES, and MCP-3. These differences on vMIP-II may be a consequence of its broad-range receptor recognition capabilities.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Anti-HIV Agents / chemistry*
  • Chemokine CCL11
  • Chemokine CCL5 / chemistry*
  • Chemokine CCL7
  • Chemokines / chemistry*
  • Chemokines, CC / chemistry*
  • Chemotactic Factors, Eosinophil / chemistry*
  • Crystallography, X-Ray
  • Cytokines / chemistry*
  • Herpesvirus 8, Human / metabolism
  • Humans
  • Models, Molecular
  • Molecular Sequence Data
  • Monocyte Chemoattractant Proteins / chemistry*
  • Receptors, CCR3
  • Receptors, Chemokine / metabolism*
  • Receptors, Virus / metabolism
  • Sequence Alignment
  • Sequence Homology, Amino Acid

Substances

  • Anti-HIV Agents
  • CCL11 protein, human
  • CCL7 protein, human
  • CCR3 protein, human
  • Chemokine CCL11
  • Chemokine CCL5
  • Chemokine CCL7
  • Chemokines
  • Chemokines, CC
  • Chemotactic Factors, Eosinophil
  • Cytokines
  • Monocyte Chemoattractant Proteins
  • Receptors, CCR3
  • Receptors, Chemokine
  • Receptors, Virus
  • vMIP-II

Associated data

  • PDB/1CM9