Onset of bronchodilation of budesonide/formoterol vs. salmeterol/fluticasone in single inhalers

Pulm Pharmacol Ther. 2001;14(1):29-34. doi: 10.1006/pupt.2000.0260.

Abstract

Combinations of inhaled glucocorticoids and long-acting beta2-agonists in the same inhaler device have become available in recent years. In this double-blind, randomized, placebo-controlled and crossover study we have evaluated the onset of action of budesonide and formoterol in a single inhaler (Symbicort Turbuhaler) and that of the fixed combination of salmeterol and fluticasone (Seretide Diskus). Thirty patients with a mean FEV1 of 2.54 l (range: 1.48-4.28) and a mean inclusion reversibility in FEV1 of 19.1% were included. Single doses of budesonide/formoterol 160/4.5 microg and 2x (160/4.5) microg, salmeterol/fluticasone 50/250 microg, or placebo were given. Serial measurements of FEV1 were performed over 3 h. The combination of one or two inhalations of budesonide/formoterol showed a faster onset of action than salmeterol/fluticasone, both evaluated as mean FEV1 at 3 min (2.74, 2.75 and 2.56 l respectively P<0.001 for both doses of budesonide/formoterol), or as average FEV1 from 0 to 15 min (2.80, 2.83 and 2.67 l respectively P<0.001 for both doses of budesonide/formoterol). For placebo, mean FEV1 at 3 min was 2.46 l, and the average FEV1 at 0-15 min was 2.50 l. Furthermore, budesonide/formoterol at both doses resulted in higher FEV1 than salmeterol/fluticasone at 3 h. We conclude that the combination of budesonide/formoterol has a faster onset of action than salmeterol/fluticasone.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Administration, Inhalation
  • Adult
  • Aged
  • Albuterol / administration & dosage
  • Albuterol / analogs & derivatives*
  • Albuterol / pharmacology*
  • Androstadienes / administration & dosage
  • Androstadienes / pharmacology*
  • Asthma / drug therapy*
  • Asthma / pathology
  • Bronchodilator Agents / administration & dosage
  • Bronchodilator Agents / pharmacology*
  • Budesonide / administration & dosage
  • Budesonide / pharmacology*
  • Cross-Over Studies
  • Double-Blind Method
  • Drug Therapy, Combination
  • Ethanolamines / administration & dosage
  • Ethanolamines / pharmacology*
  • Female
  • Fluticasone
  • Forced Expiratory Volume
  • Formoterol Fumarate
  • Humans
  • Male
  • Middle Aged
  • Salmeterol Xinafoate
  • Spirometry
  • Treatment Outcome

Substances

  • Androstadienes
  • Bronchodilator Agents
  • Ethanolamines
  • Budesonide
  • Salmeterol Xinafoate
  • Fluticasone
  • Albuterol
  • Formoterol Fumarate