Effects of Shilajit on the development of tolerance to morphine in mice

Phytother Res. 2001 Mar;15(2):177-9. doi: 10.1002/ptr.857.

Abstract

Effects of concomitant administration of Processed Shilajit (PS, 0.1 and 1 mg/kg, i.p.), in Swiss mice were evaluated on the development of tolerance to morphine induced analgesia in the hot plate test. Chronic administration of morphine (10 mg/kg, i.p., b.i.d.) to mice over a duration of 10 days resulted in the development of tolerance to the analgesic effect of morphine. Concomitant administration of PS with morphine, from day 6 to day 10, resulted in a significant inhibition of the development of tolerance to morphine (10 mg/kg, i.p.) induced analgesia. Processed Shilajit per se, in the doses used, did not elicit any significant analgesia in mice; nor did the chronic concomitant administration of Processed Shilajit alter the morphine-induced analgesia. These findings with Processed Shilajit indicate its potential as a prospective modifier of analgesic tolerance to morphine.

MeSH terms

  • Analgesics / pharmacokinetics*
  • Analgesics / therapeutic use*
  • Animals
  • Area Under Curve
  • Drug Synergism
  • Drug Tolerance
  • Female
  • Male
  • Mice
  • Morphine / pharmacokinetics*
  • Pain / prevention & control*
  • Plant Extracts / pharmacokinetics*
  • Plant Extracts / therapeutic use*
  • Plants, Medicinal*

Substances

  • Analgesics
  • Plant Extracts
  • Morphine