T-loop phosphorylation stabilizes the CDK7-cyclin H-MAT1 complex in vivo and regulates its CTD kinase activity

EMBO J. 2001 Jul 16;20(14):3749-59. doi: 10.1093/emboj/20.14.3749.

Abstract

Cyclin-dependent kinase (CDK)7-cyclin H, the CDK-activating kinase (CAK) and TFIIH-associated kinase in metazoans can be activated in vitro through T-loop phosphorylation or binding to the RING finger protein MAT1. Although the two mechanisms can operate independently, we show that in a physiological setting, MAT1 binding and T-loop phosphorylation cooperate to stabilize the CAK complex of Drosophila. CDK7 forms a stable complex with cyclin H and MAT1 in vivo only when phosphorylated on either one of two residues (Ser164 or Thr170) in its T-loop. Mutation of both phosphorylation sites causes temperature-dependent dissociation of CDK7 complexes and lethality. Furthermore, phosphorylation of Thr170 greatly stimulates the activity of the CDK7- cyclin H-MAT1 complex towards the C-terminal domain of RNA polymerase II without significantly affecting activity towards CDK2. Remarkably, the substrate-specific increase in activity caused by T-loop phosphorylation is due entirely to accelerated enzyme turnover. Thus phosphorylation on Thr170 could provide a mechanism to augment CTD phosphorylation by TFIIH-associated CDK7, and thereby regulate transcription.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Biopolymers
  • Cyclin H
  • Cyclin-Dependent Kinase-Activating Kinase
  • Cyclin-Dependent Kinases*
  • Cyclins / antagonists & inhibitors
  • Cyclins / metabolism*
  • Drosophila
  • Drosophila Proteins
  • Kinetics
  • Molecular Sequence Data
  • Phosphorylation
  • Protein Kinases / metabolism*
  • Protein Serine-Threonine Kinases / antagonists & inhibitors
  • Protein Serine-Threonine Kinases / metabolism*
  • Substrate Specificity

Substances

  • Biopolymers
  • CycH protein, Drosophila
  • Cyclin H
  • Cyclins
  • Drosophila Proteins
  • Protein Kinases
  • carboxy-terminal domain kinase
  • Protein Serine-Threonine Kinases
  • Cyclin-Dependent Kinases
  • Cyclin-Dependent Kinase-Activating Kinase