Chronic ethanol consumption impairs adrenoceptor- and purinoceptor-mediated relaxations of isolated rat detrusor smooth muscle

BJU Int. 2001 Aug;88(3):278-83. doi: 10.1046/j.1464-410x.2001.02270.x.

Abstract

Objective: To investigate the effects of chronic ethanol consumption on the reactivity of detrusor smooth muscle.

Materials and methods: Eight male rats received ethanol (7.2% v/v) in a modified liquid diet for 4 weeks. Two control groups were assessed; eight rats in one group were fed sucrose and received a liquid diet, and 12 rats in the second group received standard rat chow and water for 4 weeks. The reactivity of detrusor smooth muscle strips from ethanol-fed animals and control animals was evaluated in organ chambers.

Results: The relaxation response elicited by isoprenaline or adenosine was unaffected in the both control groups while it was significantly inhibited, with decreased maximum responses and pD2 values, in the ethanol-fed group. Contractile responses of detrusor smooth muscle to carbachol or 80 mmol/L KCl and relaxant responses to papaverine were similar in the control groups and the ethanol-fed group. There was no change in agonist potency among the groups.

Conclusion: Chronic ethanol consumption impairs beta-adrenoceptor- and purinoceptor-mediated relaxation but not cholinoceptor-mediated contraction of the rat detrusor smooth muscle. Thus, it appears that different regulatory mechanisms are involved in ethanol-induced alterations in beta-adrenergic, purinergic and muscarinic receptors in detrusor strip.

MeSH terms

  • Adenosine / pharmacology
  • Alcohol Drinking / adverse effects*
  • Animals
  • Carbachol / pharmacology
  • Dose-Response Relationship, Drug
  • Ethanol / blood
  • Ethanol / pharmacology
  • Isoproterenol / pharmacology
  • Male
  • Muscle Relaxation / drug effects*
  • Muscle, Smooth / drug effects*
  • Papaverine / pharmacology
  • Rats
  • Rats, Wistar
  • Receptors, Adrenergic, beta / drug effects*
  • Receptors, Purinergic / drug effects*

Substances

  • Receptors, Adrenergic, beta
  • Receptors, Purinergic
  • Ethanol
  • Carbachol
  • Papaverine
  • Adenosine
  • Isoproterenol