Membrane targeting of C2 domains of phospholipase C-delta isoforms

J Biol Chem. 2002 Feb 1;277(5):3568-75. doi: 10.1074/jbc.M109705200. Epub 2001 Nov 12.

Abstract

The C2 domain is a Ca(2+)-dependent membrane-targeting module found in many cellular proteins involved in signal transduction or membrane trafficking. To understand the mechanisms by which the C2 domain mediates the membrane targeting of PLC-delta isoforms, we measured the in vitro membrane binding of the C2 domains of PLC-delta1, -delta3, and -delta4 by surface plasmon resonance and monolayer techniques and their subcellular localization by time-lapse confocal microscopy. The membrane binding of the PLC-delta1-C2 is driven by nonspecific electrostatic interactions between the Ca(2+)-induced cationic surface of protein and the anionic membrane and specific interactions involving Ca(2+), Asn(647), and phosphatidylserine (PS). The PS selectivity of PLC-delta1-C2 governs its specific Ca(2+)-dependent subcellular targeting to the plasma membrane. The membrane binding of the PLC-delta3-C2 also involves Ca(2+)-induced nonspecific electrostatic interactions and PS coordination, and the latter leads to specific subcellular targeting to the plasma membrane. In contrast to PLC-delta1-C2 and PLC-delta3-C2, PLC-delta4-C2 has significant Ca(2+)-independent membrane affinity and no PS selectivity due to the presence of cationic residues in the Ca(2+)-binding loops and the substitution of Ser for the Ca(2+)-coordinating Asp in position 717. Consequently, PLC-delta4-C2 exhibits unique pre-localization to the plasma membrane prior to Ca(2+) import and non-selective Ca(2+)-mediated targeting to various cellular membranes, suggesting that PLC-delta4 might have a novel regulatory mechanism. Together, these results establish the C2 domains of PLC-delta isoforms as Ca(2+)-dependent membrane targeting domains that have distinct membrane binding properties that control their subcellular localization behaviors.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Aspartic Acid
  • Binding Sites
  • Calcium / metabolism
  • Calcium / pharmacology
  • Catalytic Domain
  • Cell Line
  • Genetic Vectors
  • Glutathione Transferase / genetics
  • Humans
  • Isoenzymes / chemistry*
  • Isoenzymes / genetics
  • Isoenzymes / metabolism
  • Kinetics
  • Models, Molecular
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Phosphatidylcholines / metabolism
  • Phospholipase C delta
  • Polymerase Chain Reaction
  • Protein Conformation
  • Protein Isoforms
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism
  • Sequence Alignment
  • Sequence Homology, Amino Acid
  • Subcellular Fractions / enzymology
  • Surface Plasmon Resonance
  • Transfection
  • Type C Phospholipases / chemistry*
  • Type C Phospholipases / genetics
  • Type C Phospholipases / metabolism

Substances

  • Isoenzymes
  • Phosphatidylcholines
  • Protein Isoforms
  • Recombinant Proteins
  • Aspartic Acid
  • Glutathione Transferase
  • Type C Phospholipases
  • PLCD1 protein, human
  • PLCD3 protein, human
  • PLCD4 protein, human
  • Phospholipase C delta
  • Calcium