In vitro and in vivo evaluation of aminopeptidase inhibitors as antimicrosporidial therapies

J Eukaryot Microbiol. 2001:Suppl:95S-98S. doi: 10.1111/j.1550-7408.2001.tb00468.x.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Aminopeptidases / antagonists & inhibitors*
  • Animals
  • Anti-Bacterial Agents / pharmacology
  • Cyclohexanes
  • Disease Models, Animal
  • Encephalitozoon cuniculi / drug effects*
  • Encephalitozoon cuniculi / growth & development
  • Encephalitozoonosis / drug therapy*
  • Encephalitozoonosis / mortality*
  • Encephalitozoonosis / parasitology
  • Enzyme Inhibitors / pharmacology*
  • Enzyme Inhibitors / therapeutic use*
  • Fatty Acids, Unsaturated / pharmacology
  • Female
  • Leucine / analogs & derivatives*
  • Leucine / pharmacology
  • Leucine / therapeutic use
  • Mice
  • Mice, Nude
  • O-(Chloroacetylcarbamoyl)fumagillol
  • Parasitic Sensitivity Tests / methods
  • Peptides*
  • Sesquiterpenes / pharmacology
  • Sesquiterpenes / therapeutic use

Substances

  • Anti-Bacterial Agents
  • Cyclohexanes
  • Enzyme Inhibitors
  • Fatty Acids, Unsaturated
  • Peptides
  • Sesquiterpenes
  • nitrobestatin
  • amastatin
  • fumagillin
  • Aminopeptidases
  • Leucine
  • ubenimex
  • O-(Chloroacetylcarbamoyl)fumagillol