The low conductance K(+) channel in human colonic crypt cells has a voltage-dependent permeability not affected by Mg(++)

Life Sci. 2002 Jul 12;71(8):855-64. doi: 10.1016/s0024-3205(02)01638-7.

Abstract

The low conductance K(+) channel found in human colonocytes was investigated using the patch-clamp technique. The channel is Ca(++)-dependent and is blocked by Ba(++) (5 mM) with a decrease in open probability from 0.42 to 0.19. At -40 mV the slope conductance was 29 pS (using intracellular solution in the pipette). In inside-out patches, inward rectification was seen both with KCl (pipette)/NaCl (bath) solutions as well as KCl/KCl solutions. The rectification could not be affected by omitting Mg(++) from the pipette or the bath solution, neither by exposing the patches to the polyamine spermine (1 mM). Using the Goldman-Hodgkin-Katz equation we show that the permeability decreased in a linear fashion from approximately 5.2 x 10(-14) cm(3)/s to 1.8 x 10(-14) cm(3)/s (-100 to +100 mV), both with and without Mg(++) in the solutions. There was no significant difference in the nominal values of permeability. This property of the K(+) channel may facilitate the hyperpolarization needed to sustain a chloride secretion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biopsy
  • Cell Membrane / metabolism
  • Cell Membrane Permeability / drug effects
  • Colon / cytology
  • Colon / metabolism*
  • Colon / physiology
  • Colonic Diseases, Functional / pathology
  • Electrophysiology
  • Extracellular Space / metabolism
  • Humans
  • Magnesium / pharmacology*
  • Patch-Clamp Techniques
  • Potassium Channels / metabolism*
  • Potassium Channels, Calcium-Activated*
  • Potassium Channels, Inwardly Rectifying / metabolism
  • Potassium Chloride / pharmacology
  • Small-Conductance Calcium-Activated Potassium Channels

Substances

  • Potassium Channels
  • Potassium Channels, Calcium-Activated
  • Potassium Channels, Inwardly Rectifying
  • Small-Conductance Calcium-Activated Potassium Channels
  • Potassium Chloride
  • Magnesium