The interdomain region of dengue NS5 protein that binds to the viral helicase NS3 contains independently functional importin beta 1 and importin alpha/beta-recognized nuclear localization signals

J Biol Chem. 2002 Sep 27;277(39):36399-407. doi: 10.1074/jbc.M204977200. Epub 2002 Jun 24.

Abstract

Dengue virus NS5 protein is a multifunctional RNA-dependent RNA polymerase that is essential for virus replication. We have shown previously that the 37- amino acid interdomain spacer sequence (residues (369)X(2)KKX(14)KKKX(11)RKX(3)405) of Dengue2 NS5 contains a functional nuclear localization signal (NLS). In this study, beta-galactosidase fusion proteins carrying point mutations of the positively charged residues or truncations of the interdomain linker region (residues 369-389 or residues 386-405) were analyzed for nuclear import and importin binding activities to show that the N-terminal part of the linker region (residues 369-389, a/bNLS) is critical for nuclear localization and is recognized with high affinity by the conventional NLS-binding importin alpha/beta heterodimeric nuclear import receptor. We also show that the importin beta-binding site (residues 320-368, bNLS) adjacent to the a/bNLS, previously identified by yeast two-hybrid analysis, is functional as an NLS, recognized with high affinity by importin beta, and able to target beta-galactosidase to the nucleus. Intriguingly, the bNLS is highly conserved among Dengue and related flaviviruses, implying a general role for the region and importin beta in the infectious cycle.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Carcinoma, Hepatocellular / metabolism
  • Cell Nucleus / metabolism
  • Dengue Virus / metabolism*
  • Dimerization
  • Dose-Response Relationship, Drug
  • Enzyme-Linked Immunosorbent Assay
  • Fluorescent Dyes / pharmacology
  • Glutathione Transferase / metabolism
  • Kinetics
  • Microscopy, Fluorescence
  • Models, Molecular
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Nuclear Localization Signals
  • Plasmids / metabolism
  • Point Mutation
  • Protein Binding
  • Protein Structure, Tertiary
  • RNA Helicases
  • Rats
  • Recombinant Fusion Proteins / metabolism
  • Sequence Homology, Amino Acid
  • Serine Endopeptidases
  • Time Factors
  • Tumor Cells, Cultured
  • Two-Hybrid System Techniques
  • Viral Nonstructural Proteins / chemistry*
  • Viral Nonstructural Proteins / metabolism
  • alpha Karyopherins / metabolism*
  • beta Karyopherins / metabolism*
  • beta-Galactosidase / metabolism

Substances

  • Fluorescent Dyes
  • NS3 protein, flavivirus
  • NS5 protein, flavivirus
  • Nuclear Localization Signals
  • Recombinant Fusion Proteins
  • Viral Nonstructural Proteins
  • alpha Karyopherins
  • beta Karyopherins
  • Glutathione Transferase
  • beta-Galactosidase
  • Serine Endopeptidases
  • RNA Helicases