Influence of raloxifene on the efficacy of an estradiol-releasing ring for treating vaginal atrophy in postmenopausal women

Menopause. 2003 Jan-Feb;10(1):45-52. doi: 10.1097/00042192-200310010-00008.

Abstract

Objective: To determine the potential interaction of oral raloxifene 60 mg/day on the efficacy of a low-dose, estradiol-releasing vaginal ring used to treat signs and symptoms of vaginal atrophy in postmenopausal women.

Design: Randomized, double-blind, placebo-controlled, parallel treatment trial of raloxifene and placebo with open-label 17beta-estradiol ring. At 10 sites in the United States, 91 postmenopausal women with at least two signs of vaginal atrophy were treated with a 17beta-estradiol ring and randomized to receive concomitant raloxifene 60 mg/day or placebo for 6 months. Efficacy of treatments was evaluated by comparing investigator assessments of genitourinary atrophic signs, vaginal maturation value, and participant assessments of vaginal symptoms at 6 months. Other measures included rate and severity of hot flashes and assessment of sexual function. Uterine safety was assessed by endometrial biopsy and transvaginal ultrasound.

Results: In women treated with a 17beta-estradiol ring, both the raloxifene and placebo treatment groups showed improvements in signs and symptoms of vaginal atrophy at 6 months, with no significant differences in degree of improvement between groups. There were no signs of endometrial proliferation in either group.

Conclusions: Concomitant administration of raloxifene does not alter the effects of the 17beta-estradiol ring on alleviating signs and symptoms of genitourinary atrophy in postmenopausal women.

Publication types

  • Clinical Trial
  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Intravaginal
  • Administration, Oral
  • Adult
  • Aged
  • Aged, 80 and over
  • Atrophy / drug therapy
  • Atrophy / pathology
  • Double-Blind Method
  • Estradiol / administration & dosage
  • Estradiol / therapeutic use*
  • Estrogen Antagonists / administration & dosage
  • Estrogen Antagonists / pharmacology*
  • Female
  • Hot Flashes / drug therapy*
  • Hot Flashes / pathology
  • Humans
  • Middle Aged
  • Pessaries
  • Postmenopause*
  • Raloxifene Hydrochloride / administration & dosage
  • Raloxifene Hydrochloride / pharmacology*
  • Severity of Illness Index
  • Sexuality
  • Surveys and Questionnaires
  • Treatment Outcome
  • United States
  • Vagina / pathology*

Substances

  • Estrogen Antagonists
  • Raloxifene Hydrochloride
  • Estradiol