Reduced social interaction following 3,4-methylenedioxymethamphetamine is not associated with enhanced 5-HT 2C receptor responsivity

Neuropharmacology. 2003 Mar;44(4):439-48. doi: 10.1016/s0028-3908(02)00407-0.

Abstract

This study examined the long-term change in serotonergic (5-hydroxytryptamine, 5-HT) neuronal function and 5-HT(2C) receptor agonist-induced behaviour following treatment of young rats with 3,4-methylenedioxymethamphetamine (MDMA). On post-natal day (PND) 28, Lister-hooded rats received either MDMA (15 mg/kg i.p.) or saline (1 ml/kg i.p.) twice daily for 3 days. On PND 50 social interaction was assessed between treatment-matched pairs of rats derived from separate litters. The effect of either the 5-HT(2C) receptor agonist, m-chlorophenylpiperazine (m-CPP, 2.5 or 1 mg/kg i.p., respectively) or saline was examined on open-field exploration (PND 52) and elevated plus-maze behaviour (PND 56). Acutely, MDMA produced hyperlocomotion and hypothermia compared with saline injection (p<0.001). Following 20 days abstinence, social interaction was decreased by 26% (p<0.05) in MDMA pre-treated rats compared with saline controls, without any change in locomotion. There was no difference in open-field or elevated plus-maze behaviour between pre-treatment groups. m-CPP caused hypolocomotion in the open-field and decreased both the percentage entries into, and time spent in, the open arms of the elevated plus-maze to a comparable extent in MDMA and saline pre-treated rats. Hippocampal and frontal cortical 5-HT and 5-hydroxyindoleacetic acid (5-HIAA) were significantly reduced in MDMA pre-treated rats, without any change in [(3)H]paroxetine binding or plasma corticosterone levels. These data suggest that the MDMA-induced reduction in social interaction is not mediated via alteration of 5-HT(2C) receptor function.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Brain / drug effects
  • Brain / metabolism
  • Corticosterone / blood
  • Exploratory Behavior / drug effects
  • Hydroxyindoleacetic Acid / metabolism
  • Hypothermia / chemically induced
  • In Vitro Techniques
  • Male
  • Maze Learning / drug effects
  • Motor Activity / drug effects
  • N-Methyl-3,4-methylenedioxyamphetamine / adverse effects*
  • Paroxetine / metabolism
  • Piperazines / pharmacology
  • Radioligand Assay
  • Rats
  • Receptor, Serotonin, 5-HT2C
  • Receptors, Serotonin / drug effects*
  • Serotonin / metabolism
  • Serotonin Agents / adverse effects*
  • Serotonin Receptor Agonists / pharmacology
  • Social Behavior*
  • Substance Withdrawal Syndrome / metabolism
  • Substance Withdrawal Syndrome / psychology

Substances

  • Piperazines
  • Receptor, Serotonin, 5-HT2C
  • Receptors, Serotonin
  • Serotonin Agents
  • Serotonin Receptor Agonists
  • Serotonin
  • Paroxetine
  • Hydroxyindoleacetic Acid
  • N-Methyl-3,4-methylenedioxyamphetamine
  • 1-(3-chlorophenyl)piperazine
  • Corticosterone