Uncompetitive antagonist binding: a biochemical index of activation of the NMDA receptor-coupled ion channel

Epilepsy Res Suppl. 1992:8:181-8. doi: 10.1016/b978-0-444-89710-7.50028-8.
No abstract available

MeSH terms

  • 2-Amino-5-phosphonovalerate / pharmacology
  • Animals
  • Binding, Competitive / drug effects
  • Binding, Competitive / physiology
  • Culture Techniques
  • Glutamates / pharmacology
  • Glutamic Acid
  • Hippocampus / drug effects*
  • Hippocampus / physiology
  • Ibotenic Acid / analogs & derivatives
  • Ibotenic Acid / pharmacology
  • Ion Channels / drug effects*
  • Ion Channels / physiology
  • Kainic Acid / pharmacology
  • N-Methylaspartate / pharmacology
  • N-Methylaspartate / physiology*
  • Phencyclidine / analogs & derivatives*
  • Phencyclidine / pharmacokinetics
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, N-Methyl-D-Aspartate / drug effects*
  • Receptors, N-Methyl-D-Aspartate / physiology
  • Synaptic Transmission / drug effects*
  • Synaptic Transmission / physiology
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid

Substances

  • Glutamates
  • Ion Channels
  • Receptors, N-Methyl-D-Aspartate
  • Ibotenic Acid
  • Glutamic Acid
  • N-Methylaspartate
  • 2-Amino-5-phosphonovalerate
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid
  • tenocyclidine
  • Phencyclidine
  • Kainic Acid