Novel players in pancreatic islet signaling: from membrane receptors to nuclear channels

Diabetes. 2004 Feb:53 Suppl 1:S86-91. doi: 10.2337/diabetes.53.2007.s86.

Abstract

Glucose and other nutrients regulate many aspects of pancreatic islet physiology. This includes not only insulin release, but also insulin synthesis and storage and other aspects of beta-cell biology, including cell proliferation, apoptosis, differentiation, and gene expression. This implies that in addition to the well-described signals for insulin release, other intracellular signaling mechanisms are needed. Here we describe the role of global and local Ca(2+) signals in insulin release, the regulation of these signals by new membrane receptors, and the generation of nuclear Ca(2+) signals involved in gene expression. An integrated view of these pathways should improve the present description of the beta-cell biology and provide new targets for novel drugs.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Gene Expression Regulation
  • Glucose / pharmacology
  • Humans
  • Ion Channels / physiology*
  • Islets of Langerhans / drug effects
  • Islets of Langerhans / physiology*
  • Models, Biological
  • Receptors, Cell Surface / physiology*
  • Receptors, Cytoplasmic and Nuclear / physiology*
  • Signal Transduction / physiology*

Substances

  • Ion Channels
  • Receptors, Cell Surface
  • Receptors, Cytoplasmic and Nuclear
  • Glucose