RyR2 and calpain-10 delineate a novel apoptosis pathway in pancreatic islets

J Biol Chem. 2004 Jun 4;279(23):24794-802. doi: 10.1074/jbc.M401216200. Epub 2004 Mar 25.

Abstract

Cells are programmed to die when critical signaling and metabolic pathways are disrupted. Inhibiting the type 2 ryanodine receptor (RyR2) in human and mouse pancreatic beta-cells markedly increased apoptosis. This mode of programmed cell death was not associated with robust caspase-3 activation prompting a search for an alternative mechanism. Increased calpain activity and calpain gene expression suggested a role for a calpain-dependent death pathway. Using a combination of pharmacological and genetic approaches, we demonstrated that the calpain-10 isoform mediated ryanodine-induced apoptosis. Apoptosis induced by the fatty acid palmitate and by low glucose also required calpain-10. Ryanodine-induced calpain activation and apoptosis were reversed by glucagon-like peptide or short-term exposure to high glucose. Thus RyR2 activity seems to play an essential role in beta-cell survival in vitro by suppressing a death pathway mediated by calpain-10, a type 2 diabetes susceptibility gene with previously unknown function.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Apoptosis*
  • Calcium / metabolism
  • Calpain / metabolism
  • Calpain / physiology*
  • Caspase 3
  • Caspases / metabolism
  • Cell Survival
  • Dantrolene / metabolism
  • Enzyme Activation
  • Gene Expression Regulation
  • Glucagon-Like Peptides
  • Glucose / metabolism
  • Humans
  • Islets of Langerhans / metabolism
  • Islets of Langerhans / pathology*
  • Mice
  • Mice, Knockout
  • Mice, Transgenic
  • Microscopy, Confocal
  • Microscopy, Fluorescence
  • Models, Biological
  • Palmitic Acids / chemistry
  • Peptides / pharmacology
  • Protein Isoforms
  • RNA, Messenger / metabolism
  • Ryanodine / metabolism
  • Ryanodine Receptor Calcium Release Channel / physiology*
  • Time Factors

Substances

  • Palmitic Acids
  • Peptides
  • Protein Isoforms
  • RNA, Messenger
  • Ryanodine Receptor Calcium Release Channel
  • Ryanodine
  • Glucagon-Like Peptides
  • glucagon-like-immunoreactivity
  • CASP3 protein, human
  • Calpain
  • Casp3 protein, mouse
  • Caspase 3
  • Caspases
  • calpain 10
  • Dantrolene
  • Glucose
  • Calcium