A novel phosphoglucose isomerase (PGI)/phosphomannose isomerase from the crenarchaeon Pyrobaculum aerophilum is a member of the PGI superfamily: structural evidence at 1.16-A resolution

J Biol Chem. 2004 Sep 17;279(38):39838-45. doi: 10.1074/jbc.M406855200. Epub 2004 Jul 13.

Abstract

The crystal structure of a dual specificity phosphoglucose isomerase (PGI)/phosphomannose isomerase from Pyrobaculum aerophilum (PaPGI/PMI) has been determined in native form at 1.16-A resolution and in complex with the enzyme inhibitor 5-phosphoarabinonate at 1.45-A resolution. The similarity of its fold, with the inner core structure of PGIs from eubacterial and eukaryotic sources, confirms this enzyme as a member of the PGI superfamily. The almost total conservation of amino acids in the active site, including the glutamate base catalyst, shows that PaPGI/PMI uses the same catalytic mechanisms for both ring opening and isomerization for the interconversion of glucose 6-phosphate (Glc-6-P) to fructose 6-phosphate (Fru-6-P). The lack of structural differences between native and inhibitor-bound enzymes suggests this activity occurs without any of the conformational changes that are the hallmark of the well characterized PGI family. The lack of a suitable second base in the active site of PaPGI/PMI argues against a PMI mechanism involving a trans-enediol intermediate. Instead, PMI activity may be the result of additional space in the active site imparted by a threonine, in place of a glutamine in other PGI enzymes, which could permit rotation of the C-2-C-3 bond of mannose 6-phosphate.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Glucose-6-Phosphate Isomerase / chemistry*
  • Glucose-6-Phosphate Isomerase / metabolism*
  • Mannose-6-Phosphate Isomerase / chemistry*
  • Mannose-6-Phosphate Isomerase / metabolism*
  • Molecular Sequence Data
  • Multigene Family
  • Pentosephosphates / metabolism
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Pyrobaculum / enzymology*
  • Substrate Specificity

Substances

  • Pentosephosphates
  • arabinonate-5-phosphate
  • Mannose-6-Phosphate Isomerase
  • Glucose-6-Phosphate Isomerase

Associated data

  • PDB/1TZB
  • PDB/1TZC