Abstract
A systematic approach through computer assisted design to identify novel quinazolines having anxiolytic and GABAergic activity has been reported.
MeSH terms
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Animals
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Anti-Anxiety Agents / chemistry*
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Anti-Anxiety Agents / pharmacology
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Dose-Response Relationship, Drug
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GABA Agents / chemistry*
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GABA Agents / pharmacology
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GABA Agonists / chemistry
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GABA Agonists / pharmacology
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GABA-A Receptor Agonists
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Maze Learning / drug effects
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Maze Learning / physiology
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Mice
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Quinazolines / chemistry*
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Quinazolines / pharmacology
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Receptors, GABA-A / physiology
Substances
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Anti-Anxiety Agents
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GABA Agents
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GABA Agonists
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GABA-A Receptor Agonists
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Quinazolines
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Receptors, GABA-A