[153Sm]EDTMP: a potential therapy for bone cancer pain

Semin Nucl Med. 1992 Jan;22(1):41-5. doi: 10.1016/s0001-2998(05)80156-4.

Abstract

Reactor-produced samarium-153 (153Sm) is both a beta and gamma emitter with a physical half-life of 46.3 hours. When complexed with EDTMP, more than 50% of the administered dose localizes in bone. A therapeutic trial on patients with painful bone metastases performed at the University of Missouri produced relief in 65.4% of the patients who were evaluable. Myelotoxicity was mild and transient. For [153Sm]EDTMP to attain clinical utility, studies demonstrating its efficacy as an analgesic must be performed to exclude a "ligand analgesic effect".

Publication types

  • Review

MeSH terms

  • Animals
  • Bone Neoplasms / physiopathology
  • Bone Neoplasms / secondary*
  • Dogs
  • Humans
  • Neoplasms / etiology
  • Neoplasms / radiotherapy*
  • Organometallic Compounds / therapeutic use*
  • Organophosphorus Compounds / therapeutic use*

Substances

  • Organometallic Compounds
  • Organophosphorus Compounds
  • samarium Sm-153 lexidronam