Abstract
Intracellular photolysis of a novel 'caged' capsaicin analogue results in in vitro activation of the capsaicin receptor TRPV1.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Animals
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Calcium / metabolism
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Capsaicin / analogs & derivatives*
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Cells, Cultured
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Diterpenes / pharmacology
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Electrophysiology
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Humans
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Ion Channels / metabolism
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Light
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Models, Chemical
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Neurons / metabolism
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Protein Binding
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Rats
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Structure-Activity Relationship
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TRPV Cation Channels / antagonists & inhibitors*
Substances
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Diterpenes
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Ion Channels
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TRPV Cation Channels
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TRPV1 protein, human
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Trpv1 protein, rat
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resiniferatoxin
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Capsaicin
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Calcium