Inhibition of TFII-I-dependent cell cycle regulation by p53

Mol Cell Biol. 2005 Dec;25(24):10940-52. doi: 10.1128/MCB.25.24.10940-10952.2005.

Abstract

The multifunctional transcription factor TFII-I is tyrosine phosphorylated in response to extracellular growth signals and transcriptionally activates growth-promoting genes. However, whether activation of TFII-I also directly affects the cell cycle profile is unknown. Here we show that under normal growth conditions, TFII-I is recruited to the cyclin D1 promoter and transcriptionally activates this gene. Most strikingly, upon cell cycle arrest resulting from genotoxic stress and p53 activation, TFII-I is ubiquitinated and targeted for proteasomal degradation in a p53- and ATM (ataxia telangiectasia mutated)-dependent manner. Consistent with a direct role of TFII-I in cell cycle regulation and cellular proliferation, stable and ectopic expression of wild-type TFII-I increases cyclin D1 levels, resulting in accelerated entry to and exit from S phase, and overcomes p53-mediated cell cycle arrest, despite radiation. We further show that the transcriptional regulation of cyclin D1 and cell cycle control by TFII-I are dependent on its tyrosine phosphorylation at positions 248 and 611, sites required for its growth signal-mediated transcriptional activity. Taken together, our data define TFII-I as a growth signal-dependent transcriptional activator that is critical for cell cycle control and proliferation and further reveal that genotoxic stress-induced degradation of TFII-I results in cell cycle arrest.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Ataxia Telangiectasia Mutated Proteins
  • Cell Cycle Proteins / metabolism
  • Cell Cycle* / genetics
  • Cell Cycle* / radiation effects
  • Cyclin D1 / genetics*
  • Cyclin D1 / metabolism
  • DNA-Binding Proteins / metabolism
  • Gamma Rays
  • Humans
  • Mice
  • NIH 3T3 Cells
  • Promoter Regions, Genetic
  • Proteasome Endopeptidase Complex / metabolism
  • Protein Serine-Threonine Kinases / metabolism
  • Transcription Factors, TFII / antagonists & inhibitors
  • Transcription Factors, TFII / genetics
  • Transcription Factors, TFII / metabolism*
  • Transcriptional Activation*
  • Tumor Suppressor Protein p53 / metabolism*
  • Tumor Suppressor Proteins / metabolism
  • Ubiquitins / metabolism

Substances

  • Cell Cycle Proteins
  • DNA-Binding Proteins
  • GTF2I protein, human
  • Transcription Factors, TFII
  • Tumor Suppressor Protein p53
  • Tumor Suppressor Proteins
  • Ubiquitins
  • Cyclin D1
  • ATM protein, human
  • Ataxia Telangiectasia Mutated Proteins
  • Atm protein, mouse
  • Protein Serine-Threonine Kinases
  • Proteasome Endopeptidase Complex