The protein phosphatase 2A represents a novel cellular target for hepatitis C virus NS5A protein

Biochimie. 2006 Jun;88(6):651-62. doi: 10.1016/j.biochi.2005.12.003. Epub 2006 Jan 18.

Abstract

It is well established that HCV NS5A protein when expressed in mammalian cells perturbs the extracellular signal regulated kinase (ERK) pathway. The protein serine/threonine phosphatase 2A controls the phosphorylation of numerous proteins involved in cell signaling and one characterized function is the regulation of Ras-Raf mitogen activated protein (MAP) kinase signaling pathways. Our results showed that expression of HCV NS5A protein stimulates phosphatase 2A (PP2A) activity in cells, indicating the relevance of NS5A as a regulator of PP2A in vivo. We found that transient expression of the full length NS5A protein in different cell lines leads to a significant increase of the PP2A activity and this activity is specifically inhibited by the addition of okadaic acid, a PP2A inhibitor, in living cells. Further investigation showed that NS5A protein interacts in vivo and in vitro with the scaffolding A and the catalytic C subunits of PP2A. We propose that HCV NS5A represents a viral PP2A regulatory protein. This is a novel function for the NS5A protein which may have a key role in the ability of the virus to deregulate cell growth and survival.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line
  • Dose-Response Relationship, Drug
  • Enzyme Activation
  • Haplorhini
  • Hepacivirus / metabolism*
  • Humans
  • Liver / cytology
  • Phosphoprotein Phosphatases / metabolism*
  • Protein Phosphatase 2
  • Protein Subunits / metabolism
  • Substrate Specificity
  • Viral Nonstructural Proteins / metabolism*

Substances

  • Protein Subunits
  • Viral Nonstructural Proteins
  • NS-5 protein, hepatitis C virus
  • Phosphoprotein Phosphatases
  • Protein Phosphatase 2