Diacerhein versus glucosamine in a rat model of osteoarthritis

Clinics (Sao Paulo). 2006 Oct;61(5):461-6. doi: 10.1590/s1807-59322006000500014.

Abstract

Purpose: The purpose of this study was to compare the chondroprotective effect of diacerein and glucosamine regarding degenerative changes and articular stiffness in an experimental model of arthritis.

Methods: Twenty rats underwent medial meniscectomy on the right knee. Ten animals were given diacerhein, and 10 were given glucosamine, from day 1 to the third month postoperatively, when all of them were killed. Histological and functional analysis of the knees were performed (measurement of maximum extension).

Results: All operated knees showed more limited extension values and more degenerative changes as compared to nonoperated contralateral sides. A comparison of the two drugs showed that the degree of articular stiffness was significantly lower with diacerein, although degenerative changes were similar.

Conclusions: 1) Prophylactic use of diacerein leads to lower degree of articular stiffness when compared to glucosamine; 2) The prophylactic chondroprotective effects of diacerein and glucosamine are histologically similar.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Anthraquinones / therapeutic use*
  • Anti-Inflammatory Agents, Non-Steroidal / therapeutic use*
  • Disease Models, Animal
  • Glucosamine / therapeutic use*
  • Male
  • Menisci, Tibial / drug effects
  • Menisci, Tibial / surgery
  • Menisci, Tibial / ultrastructure
  • Osteoarthritis, Knee / drug therapy*
  • Osteoarthritis, Knee / surgery
  • Postoperative Care
  • Rats
  • Rats, Wistar
  • Severity of Illness Index
  • Stifle / drug effects*
  • Stifle / surgery
  • Stifle / ultrastructure

Substances

  • Anthraquinones
  • Anti-Inflammatory Agents, Non-Steroidal
  • diacerein
  • Glucosamine