Isolation of neurotoxic peptides from the venom of the 'armed' spider Phoneutria nigriventer

Toxicon. 1991;29(10):1225-33. doi: 10.1016/0041-0101(91)90195-w.

Abstract

Three neurotoxic fractions, lethal to mice, were isolated from the venom of the spider Phoneutria nigriventer, by gel filtration and reverse phase chromatography (Phoneutria toxins 1, 2 and 3). These toxins have mol. wts in the range 6000-9000, and have different amino acid compositions and N-terminal amino acid sequences. The toxins also differ in the lethality and signs they cause in mice after intracerebro-ventricular injection. The median LD50 being respectively for the whole venom, toxins 1, 2 and 3, 47 +/- 5 micrograms, 45 +/- 4 micrograms, 1.7 +/- 0.7 micrograms and 137 +/- 10 micrograms/kg mouse. Toxins 1 and 2 induce excitatory symptoms in mice and toxin 3 a flaccid paralysis with an ED50 of 40 +/- 5 micrograms/kg mouse as measured also by intracerebro-ventricular injection. The presence in the venom of a non-neurotoxic, smooth muscle active peptide is also described.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Amino Acids / analysis
  • Animals
  • Chromatography, Gel
  • Chromatography, Liquid
  • Female
  • Guinea Pigs
  • Injections, Intraventricular
  • Lethal Dose 50
  • Mice
  • Molecular Sequence Data
  • Molecular Weight
  • Muscle Contraction / drug effects
  • Muscle, Smooth / drug effects
  • Neurotoxins / analysis
  • Neurotoxins / isolation & purification*
  • Neurotoxins / toxicity
  • Peptides / analysis
  • Peptides / isolation & purification*
  • Peptides / toxicity
  • Spider Venoms / analysis*
  • Spiders / metabolism*

Substances

  • Amino Acids
  • Neurotoxins
  • Peptides
  • Spider Venoms