GSK-3-mediated phosphorylation enhances Maf-transforming activity

Mol Cell. 2007 Nov 30;28(4):584-97. doi: 10.1016/j.molcel.2007.11.009.

Abstract

The Maf oncoproteins are b-Zip transcription factors of the AP-1 superfamily. They are involved in developmental, metabolic, and tumorigenic processes. Maf proteins are overexpressed in about 50% of human multiple myelomas. Here, we show that Maf-transforming activity is controlled by GSK-3-dependent phosphorylation and that phosphorylation by GSK-3 can increase the oncogenic activity of a protein. Using microarray analysis, we identify a gene-expression subprogram regulated by GSK-3-mediated Maf phosphorylation involved in extracellular matrix remodeling and relevant to cancer progression. We also demonstrate that GSK-3 triggers MafA sequential phosphorylation on residues S61, T57, T53, and S49, inducing its ubiquitination and degradation. Paradoxically, this phosphorylation increases MafA-transcriptional activity through the recruitment of the coactivator P/CAF. We further demonstrate that P/CAF protects MafA from ubiquitination and degradation, suggesting that, upon the release of the coactivator complex, MafA becomes polyubiquitinated and degraded to allow the response to terminate.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • COS Cells
  • Cell Line
  • Cell Transformation, Neoplastic*
  • Chickens
  • Chlorocebus aethiops
  • Glycogen Synthase Kinase 3 / metabolism*
  • Humans
  • Maf Transcription Factors, Large / chemistry
  • Maf Transcription Factors, Large / genetics
  • Maf Transcription Factors, Large / metabolism*
  • Molecular Sequence Data
  • Phosphorylation
  • Phosphoserine / metabolism
  • Phosphothreonine / metabolism
  • Protein Processing, Post-Translational
  • Rats
  • Transcription, Genetic
  • Ubiquitination
  • p300-CBP Transcription Factors / metabolism

Substances

  • Maf Transcription Factors, Large
  • Phosphothreonine
  • Phosphoserine
  • p300-CBP Transcription Factors
  • p300-CBP-associated factor
  • Glycogen Synthase Kinase 3

Associated data

  • GEO/GSE9045