The role of 5-hydroxytryptophan (5-HTP) in the regulation of the sleep/wake cycle in parachlorophenylalanine (p-CPA) pretreated rat: a multiple approach study

Exp Brain Res. 1991;86(1):117-24. doi: 10.1007/BF00231046.

Abstract

In the rat, the insomnia which follows the administration of parachlorophenylalanine (p-CPA), a serotonin synthesis inhibitor, is transiently reversed either by intra-cisternal injection of L-5-HTP or by an associated injection of 5-HTP and an L-aromatic-acid-decarboxylase inhibitor (benserazide). Histochemical, immunohistochemical and chemical investigations showed that 5-HTP administration does not lead to a detectable increase in cerebral 5-HT. These findings suggest that the restoration of sleep after p-CPA treatment could be mediated by the central action of 5-HTP.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 5-Hydroxytryptophan / administration & dosage
  • 5-Hydroxytryptophan / metabolism
  • 5-Hydroxytryptophan / physiology*
  • Animals
  • Autoradiography
  • Benserazide / pharmacology
  • Brain Chemistry / drug effects
  • Cisterna Magna
  • Fenclonine / pharmacology*
  • Immunohistochemistry
  • Injections
  • Male
  • Rats
  • Rats, Inbred Strains
  • Serotonin / metabolism
  • Sleep / drug effects
  • Sleep / physiology*

Substances

  • Serotonin
  • Benserazide
  • 5-Hydroxytryptophan
  • Fenclonine