Histone deacetylase 6 interacts with the microtubule-associated protein tau

J Neurochem. 2008 Sep;106(5):2119-30. doi: 10.1111/j.1471-4159.2008.05564.x. Epub 2008 Jul 12.

Abstract

Histone deacetylase 6 (HDAC6), a unique cytoplasmic deacetylase, likely plays a role in neurodegeneration by coordinating cell responses to abnormal protein aggregation. Here, we provide in vitro and in vivo evidence that HDAC6 interacts with tau, a microtubule-associated protein that forms neurofibrillary tangles in Alzheimer's disease. This interaction is mediated by the microtubule-binding domain on tau and the Ser/Glu tetradecapeptide domain on HDAC6. Treatment with tubacin, a selective inhibitor of tubulin deacetylation activity of HDAC6, did not disrupt HDAC6-tau interaction. Nonetheless tubacin treatment attenuated site-specific tau phosphorylation, as did shRNA-mediated knockdown of HDAC6. Proteasome inhibition potentiated HDAC6-tau interactions and facilitated the concentration and co-localization of HDAC6 and tau in a perinuclear aggresome-like compartment, independent of HDAC6 tubulin deacetylase activity. Furthermore, we observed that in Alzheimer's disease brains the protein level of HDAC6 was significantly increased. These findings establish HDAC6 as a tau-interacting protein and as a potential modulator of tau phosphorylation and accumulation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Alzheimer Disease / genetics
  • Alzheimer Disease / metabolism*
  • Anilides / pharmacology
  • Brain / metabolism*
  • Brain / pathology
  • Cell Compartmentation / physiology
  • Cell Line
  • Down-Regulation / genetics
  • Enzyme Inhibitors / pharmacology
  • Female
  • Histone Deacetylase 6
  • Histone Deacetylases / genetics
  • Histone Deacetylases / metabolism*
  • Humans
  • Hydroxamic Acids / pharmacology
  • Male
  • Microtubules / metabolism
  • Middle Aged
  • Neurofibrillary Tangles / metabolism
  • Neurofibrillary Tangles / pathology
  • Neurons / metabolism*
  • Neurons / pathology
  • Organelles / metabolism
  • Phosphorylation / drug effects
  • Protein Binding / physiology
  • Protein Structure, Tertiary / physiology
  • RNA, Small Interfering / genetics
  • tau Proteins / metabolism*

Substances

  • Anilides
  • Enzyme Inhibitors
  • Hydroxamic Acids
  • RNA, Small Interfering
  • tau Proteins
  • tubacin
  • HDAC6 protein, human
  • Histone Deacetylase 6
  • Histone Deacetylases