Effects of methylprednisolone acetate and glucosamine on proteoglycan production by equine chondrocytes in vitro

Am J Vet Res. 2008 Sep;69(9):1123-8. doi: 10.2460/ajvr.69.9.1123.

Abstract

Objective: To evaluate the effects of methylprednisolone acetate (MPA) on proteoglycan production by equine chondrocytes and to investigate whether glucosamine hydrochloride modulates these effects at clinically relevant concentrations.

Sample population: Articular cartilage with normal gross appearance from metacarpophalangeal and metatarsophalangeal joints of 8 horses (1 to 10 years of age).

Procedures: In vitro chondrocyte pellets were pretreated with glucosamine (0, 1, 10, and 100 microg/mL) for 48 hours and exposed to MPA (0, 0.05, and 0.5 mg/mL) for 24 hours. Pellets and media were assayed for proteoglycan production (Alcian blue precipitation) and proteoglycan content (dimethylmethylene blue assay), and pellets were assayed for DNA content.

Results: Methylprednisolone decreased production of proteoglycan by equine chondrocytes at both concentrations studied. Glucosamine protected proteoglycan production at all 3 concentrations studied.

Conclusions and clinical relevance: Methylprednisolone, under noninflammatory conditions present in this study, decreased production of proteoglycan by equine chondrocytes. Glucosamine had a protective effect against inhibition of proteoglycan production at all 3 concentrations studied. This suggested that glucosamine may be useful as an adjunct treatment when an intra-articular injection of a corticosteroid is indicated and that it may be efficacious at concentrations relevant to clinical use.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology*
  • Cells, Cultured
  • Chondrocytes / cytology
  • Chondrocytes / drug effects*
  • DNA / metabolism
  • Glucosamine / pharmacology*
  • Glycosaminoglycans / metabolism
  • Horses / physiology*
  • Methylprednisolone / analogs & derivatives*
  • Methylprednisolone / pharmacology
  • Methylprednisolone Acetate
  • Proteoglycans / biosynthesis*
  • Proteoglycans / metabolism

Substances

  • Anti-Inflammatory Agents
  • Glycosaminoglycans
  • Proteoglycans
  • Methylprednisolone Acetate
  • DNA
  • Glucosamine
  • Methylprednisolone