The effects of renzapride, a novel prokinetic agent, in diabetic gastroparesis

Aliment Pharmacol Ther. 1991 Apr;5(2):135-42. doi: 10.1111/j.1365-2036.1991.tb00014.x.

Abstract

Gastric emptying was measured in 9 diabetic patients with autonomic neuropathy (Group 1) and 8 normal controls (Group 2) on 4 occasions after swallowing placebo, 0.5, 1.0 or 2.0 mg of the newly developed prokinetic drug renzapride given double-blind and in random order. The liquid component of the test meal was labelled with In113m and the solid with Tc99m. Liquid emptying was uni-exponential. Solid emptying comprised an initial lag phase, followed by a linear component. Following placebo, the mean lag phase of solid emptying was 40 +/- 7 (S.E.M.) min in Group 1 and 16 +/- 2 min in Group 2 (P less than 0.01). In Group 1 subjects renzapride reduced the mean lag phase by 20-26 min at all doses (P less than 0.01). No effect was seen in Group 2. The linear rate of solid emptying was similar in both groups (0.9 +/- 0.1 and 1.0 +/- 0.2%/min) and was not altered by renzapride. Mean liquid t1/2 was similar in Groups 1 and 2 after placebo (30 +/- 6 and 29 +/- 4 min, respectively) and was decreased with increasing doses of renzapride in both groups. No adverse effects were encountered in any subjects. Renzapride may be useful in the treatment of diabetic gastroparesis.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Autonomic Nervous System Diseases / drug therapy
  • Autonomic Nervous System Diseases / physiopathology
  • Benzamides / adverse effects
  • Benzamides / therapeutic use*
  • Bridged Bicyclo Compounds / adverse effects
  • Bridged Bicyclo Compounds / therapeutic use*
  • Bridged Bicyclo Compounds, Heterocyclic*
  • Diabetic Neuropathies / drug therapy*
  • Diabetic Neuropathies / physiopathology
  • Double-Blind Method
  • Female
  • Gastric Emptying / drug effects
  • Humans
  • Male
  • Middle Aged
  • Serotonin Antagonists / adverse effects
  • Serotonin Antagonists / therapeutic use*
  • Stomach Diseases / drug therapy*
  • Stomach Diseases / etiology
  • Stomach Diseases / physiopathology

Substances

  • Benzamides
  • Bridged Bicyclo Compounds
  • Bridged Bicyclo Compounds, Heterocyclic
  • Serotonin Antagonists
  • renzapride