Beyond picomolar affinities: quantitative aspects of noncovalent and covalent binding of drugs to proteins

J Med Chem. 2009 Jan 22;52(2):225-33. doi: 10.1021/jm800498e.
No abstract available

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Absorption
  • Enzymes / metabolism
  • Pharmaceutical Preparations / metabolism*
  • Protein Binding
  • Proteins / metabolism*
  • Thermodynamics

Substances

  • Enzymes
  • Pharmaceutical Preparations
  • Proteins