Antimutagenic activity and radical scavenging activity of water infusions and phenolics from ligustrum plants leaves

Molecules. 2009 Jan 22;14(1):509-18. doi: 10.3390/molecules14010509.

Abstract

Water infusions of Ligustrum delavayanum and Ligustrum vulgare leaves and eight phenolics isolated therefrom have been assayed in vitro on ofloxacin-induced genotoxicity in the unicellular flagellate Euglena gracilis. The tested compounds luteolin, quercetin, luteolin-7-glucoside, luteolin-7-rutinoside, quercetin-3-rutinoside, apigenin-7-rutinoside, tyrosol and esculetin inhibited the mutagenic activity of ofloxacin (43 microM) in E. gracilis. Water infusions from leaves of L. delavayanum and L. vulgare showed higher antimutagenic effect (p(t) < 0.001). The activity of these samples against ofloxacin (86 microM)-induced genotoxicity was lower, but statistically significant (p(t) < 0.05), excluding the water infusion of L. delavayanum leaves (p(t) < 0.01). Efficacy of quercetin, luteolin-7-rutinoside, apigenin-7-rutinoside was insignificant. The antimutagenic effect of most phenolics we studied could be clearly ascribed to their DPPH scavenging activity, substitution patterns and lipophilicity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Bacterial Agents / metabolism
  • Anti-Bacterial Agents / pharmacology
  • Antimutagenic Agents / chemistry*
  • Antimutagenic Agents / metabolism
  • Biphenyl Compounds / chemistry
  • Euglena gracilis / drug effects
  • Euglena gracilis / genetics
  • Free Radical Scavengers / chemistry*
  • Free Radical Scavengers / metabolism
  • Hydrazines / chemistry
  • Ligustrum / chemistry*
  • Ofloxacin / metabolism
  • Ofloxacin / pharmacology
  • Phenols / chemistry*
  • Picrates
  • Plant Extracts / chemistry*
  • Plant Extracts / metabolism
  • Plant Leaves / chemistry*
  • Water

Substances

  • Anti-Bacterial Agents
  • Antimutagenic Agents
  • Biphenyl Compounds
  • Free Radical Scavengers
  • Hydrazines
  • Phenols
  • Picrates
  • Plant Extracts
  • Water
  • Ofloxacin
  • 1,1-diphenyl-2-picrylhydrazyl