Protection against amyloid beta cytotoxicity by sulforaphane: role of the proteasome

Arch Pharm Res. 2009 Jan;32(1):109-15. doi: 10.1007/s12272-009-1124-2. Epub 2009 Jan 29.

Abstract

The 26S proteasome plays a major role in degradation of abnormal proteins within the cell. The indirect antioxidant including sulforaphane (SFN) protects cells from oxidative damage by increasing the expression of Nrf2-target genes. It has been observed that the expression of multiple subunits of the proteasome was up-regulated by indirect antioxidants through the Nrf2 pathway. In the current study, the role of SFN in amyloid beta(1-42) (Abeta(1-42))-induced cytotoxicity has been investigated in murine neuroblastoma cells. Treatment with SFN protected cells from Abeta(1-42)-mediated cell death in Neuro2A and N1E 115 cells. Inhibition of proteasome activities by MG132 could abolish the protective effect of SFN against Abeta(1-42). Neuro2A cells, which were stably overexpressing the catalytic subunit of the proteasome PSMB5, showed an elevated resistance toward Abeta(1-42) toxicity compared to control cells. Furthermore, the in vitro assay demonstrated that the Abeta(1-42) peptide is degraded by the proteasome fraction. These results suggest that proteasome-inducing indirect antioxidants may facilitate the removal of the Abeta(1-42) peptide and lead to the amelioration of abnormal protein-associated etiologies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amyloid beta-Peptides / metabolism
  • Amyloid beta-Peptides / toxicity*
  • Animals
  • Antioxidants / pharmacology*
  • Cell Line, Tumor
  • Cell Survival / drug effects
  • Cysteine Proteinase Inhibitors / pharmacology
  • Cytoprotection
  • Dose-Response Relationship, Drug
  • Isothiocyanates
  • Leupeptins / pharmacology
  • Mice
  • Neuroblastoma / enzymology
  • Neuroblastoma / pathology
  • Neurons / drug effects*
  • Neurons / enzymology
  • Neurons / pathology
  • Peptide Fragments / metabolism
  • Peptide Fragments / toxicity*
  • Promoter Regions, Genetic
  • Proteasome Endopeptidase Complex / genetics
  • Proteasome Endopeptidase Complex / metabolism*
  • Proteasome Inhibitors
  • Sulfoxides
  • Thiocyanates / pharmacology*
  • Transfection
  • Up-Regulation

Substances

  • Amyloid beta-Peptides
  • Antioxidants
  • Cysteine Proteinase Inhibitors
  • Isothiocyanates
  • Leupeptins
  • Peptide Fragments
  • Proteasome Inhibitors
  • Sulfoxides
  • Thiocyanates
  • amyloid beta-protein (1-42)
  • Proteasome Endopeptidase Complex
  • Psmb5 protein, mouse
  • ATP dependent 26S protease
  • sulforaphane
  • benzyloxycarbonylleucyl-leucyl-leucine aldehyde