Anti-inflammatory activity of flower extract of Calendula officinalis Linn. and its possible mechanism of action

Indian J Exp Biol. 2009 Feb;47(2):113-20.

Abstract

Calendula officinalis flower extract possessed significant anti-inflammatory activity against carrageenan and dextran-induced acute paw edema. Oral administration of 250 and 500 mg/kg body weight Calendula extract produced significant inhibition (50.6 and 65.9% respectively) in paw edema of animals induced by carrageenan and 41.9 and 42.4% respectively with inflammation produced by dextran. In chronic anti-inflammatory model using formalin, administration of 250 and 500 mg/kg body weight Calendula extract produced an inhibition of 32.9 and 62.3% respectively compared to controls. TNF-alpha production by macrophage culture treated with lipopolysaccharide (LPS) was found to be significantly inhibited by Calendula extract. Moreover, increased levels of proinflammatory cytokines IL- 1beta, IL-6, TNF-alpha and IFN-gamma and acute phase protein, C- reactive protein (CRP) in mice produced by LPS injection were inhibited significantly by the extract. LPS induced cyclooxygenase-2 (Cox-2) levels in mice spleen were also found to be inhibited by extract treatment. The results showed that potent anti-inflammatory response of C. officinalis extract may be mediated by the inhibition of proinflammatory cytokines and Cox-2 and subsequent prostaglandin synthesis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / therapeutic use*
  • Calendula / chemistry*
  • Cell Line
  • Cell Shape / drug effects
  • Cyclooxygenase 2 / genetics
  • Cytokines / biosynthesis
  • Cytokines / blood
  • Flowers / chemistry*
  • Gene Expression / drug effects
  • Inflammation / chemically induced
  • Inflammation / drug therapy
  • Inflammation / immunology
  • Inflammation / pathology
  • Macrophages / cytology
  • Macrophages / drug effects
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Phytotherapy*
  • Plant Extracts / therapeutic use*

Substances

  • Anti-Inflammatory Agents
  • Cytokines
  • Plant Extracts
  • Ptgs2 protein, mouse
  • Cyclooxygenase 2