Interaction of loperamide with [3H]naloxone binding sites in guinea pig brain and myenteric plexus

Mol Pharmacol. 1977 May;13(3):533-40.
No abstract available

MeSH terms

  • Animals
  • Binding Sites / drug effects
  • Brain / drug effects
  • Brain / metabolism*
  • Drug Interactions
  • Electric Stimulation
  • Female
  • Guinea Pigs
  • Ileum / drug effects
  • Ileum / physiology
  • In Vitro Techniques
  • Loperamide / metabolism
  • Loperamide / pharmacology*
  • Male
  • Morphine / pharmacology
  • Muscle Contraction / drug effects
  • Muscle, Smooth / drug effects
  • Myenteric Plexus / drug effects
  • Myenteric Plexus / metabolism*
  • Naloxone / metabolism*
  • Naloxone / pharmacology
  • Piperidines / pharmacology*
  • Receptors, Opioid / drug effects
  • Receptors, Opioid / metabolism*

Substances

  • Piperidines
  • Receptors, Opioid
  • Naloxone
  • Loperamide
  • Morphine