Rapid homologous up-regulation of binding capacity of androgen receptors in intact cells

Biochem Biophys Res Commun. 1991 Nov 27;181(1):383-8. doi: 10.1016/s0006-291x(05)81430-5.

Abstract

Incubation of MCF 7 cells with 5 alpha-dihydrotestosterone (DHT) at 37 degrees C led to a 70% increase in the Bmax of androgen receptor, as compared to the values measured at 2 degrees C, without detectable changes in equilibrium dissociation constants. When MCF 7 cells were incubated with hormone at 2 degrees C, to reach steady-state levels of androgen-receptor complex, a subsequent temperature shift to 37 degrees C induced a rapid (t 1/2 = 3 min) cycloheximide-insensitive increase in DHT binding to androgen receptor. MCF 7 cell treatments at 37 degrees C either before or after incubation with DHT at 2 degrees C showed that up-regulation of binding capacity of androgen receptor could be observed only if hormone is present during incubation at physiological temperature.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Breast Neoplasms
  • Cell Line
  • Dihydrotestosterone / pharmacology*
  • Female
  • Humans
  • Kinetics
  • Receptors, Androgen / drug effects
  • Receptors, Androgen / metabolism*
  • Temperature
  • Up-Regulation*

Substances

  • Receptors, Androgen
  • Dihydrotestosterone