Clinical uses of low-dose ketamine in patients undergoing surgery

Curr Drug Targets. 2009 Aug;10(8):707-15. doi: 10.2174/138945009788982496.

Abstract

Ketamine acts mainly as a N-methyl-D-aspartate receptor (NMDAr) antagonist. Originally developed as a general anesthetic, it is now seldom employed as such in richer countries due to the relatively high risk of psychotomimetic adverse effects. Recently, low-dose regimens in the range of 0.25-0.5 mg/kg as an initial bolus followed by 50-500 kappag/kg/h have been proposed as an adjuvant for postoperative analgesia and for the reduction of exogenous opioid-induced hyperalgesia. In this review, we examine the evidence for clinical usefulness of perioperative ketamine infusion and its role in the context of general and/or regional anesthesia.

Publication types

  • Review

MeSH terms

  • Anesthesia, General
  • Anesthesia, Local
  • Anesthetics, Dissociative / administration & dosage
  • Anesthetics, Dissociative / therapeutic use*
  • Dose-Response Relationship, Drug
  • Excitatory Amino Acid Antagonists / administration & dosage
  • Excitatory Amino Acid Antagonists / therapeutic use*
  • Humans
  • Ketamine / administration & dosage
  • Ketamine / therapeutic use*
  • Pain, Postoperative / physiopathology
  • Pain, Postoperative / prevention & control

Substances

  • Anesthetics, Dissociative
  • Excitatory Amino Acid Antagonists
  • Ketamine