Mechanisms of action of acriflavine: electron microscopic study of cell wall changes induced in Staphylococcus aureus by acriflavine

Microbiol Immunol. 2009 Sep;53(9):481-6. doi: 10.1111/j.1348-0421.2009.00151.x.

Abstract

The antimicrobial action of acriflavine, a quaternary ammonium compound, on Staphylococcus aureus was studied by electron microscopic observation. The bactericidal activity of acriflavine was dose-dependent over the 4 hr of exposure time. Scanning electron micrographs showed a wavy wrinkled cell surface following treatment with acriflavine. Transmission electron micrographs showed thickened cell walls following treatment with acriflavine. Acriflavine-induced cell wall thickness seemed to affect both the peripheral and cross walls, but was reversible after treatment removal. These findings indicate that cell wall thickness is a characteristic phenotype of S. aureus exposed to acriflavine. It is therefore believed that cell wall thickness plays an important role in the mechanism of action of acriflavine.

MeSH terms

  • Acriflavine / pharmacology*
  • Anti-Bacterial Agents / pharmacology*
  • Cell Wall / drug effects
  • Cell Wall / ultrastructure*
  • Microscopy, Electron
  • Staphylococcus aureus / drug effects*
  • Staphylococcus aureus / ultrastructure

Substances

  • Anti-Bacterial Agents
  • Acriflavine