Gating in CNGA1 channels

Pflugers Arch. 2010 Mar;459(4):547-55. doi: 10.1007/s00424-009-0751-2. Epub 2009 Nov 7.

Abstract

The aminoacid sequences of CNG and K(+) channels share a significant sequence identity, and it has been suggested that these channels have a common ancestral 3D architecture. However, K(+) and CNG channels have profoundly different physiological properties: indeed, K(+) channels have a high ionic selectivity, their gating strongly depends on membrane voltage and when opened by a steady depolarizing voltage several K(+) channels inactivate, whereas CNG channels have a low ion selectivity, their gating is poorly voltage dependent, and they do not desensitize in the presence of a steady concentration of cyclic nucleotides that cause their opening. The purpose of the present review is to summarize and recapitulate functional and structural differences between K(+) and CNG channels with the aim to understand the gating mechanisms of CNG channels.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Cyclic Nucleotide-Gated Cation Channels / chemistry
  • Cyclic Nucleotide-Gated Cation Channels / genetics
  • Cyclic Nucleotide-Gated Cation Channels / metabolism*
  • Ion Channel Gating*
  • Models, Molecular
  • Molecular Sequence Data
  • Mutation
  • Potassium Channels / genetics
  • Potassium Channels / metabolism
  • Protein Conformation
  • Sequence Alignment

Substances

  • Cyclic Nucleotide-Gated Cation Channels
  • Potassium Channels