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Review

. 2010 Apr 8;53(7):2681-94.

doi: 10.1021/jm901443h.

Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto¹, Elena Ardini, Elena Casale, Mauro Angiolini

Affiliations

PMID: 20000735
DOI: 10.1021/jm901443h

Review

Through the "gatekeeper door": exploiting the active kinase conformation

Fabio Zuccotto et al. J Med Chem. 2010.

. 2010 Apr 8;53(7):2681-94.

doi: 10.1021/jm901443h.

Authors

Fabio Zuccotto¹, Elena Ardini, Elena Casale, Mauro Angiolini

Affiliation

¹ Department of Chemical Core Technologies, Nerviano Medical Sciences, Oncology, Viale Pasteur 10, Nerviano 20014, Italy. Fabio.Zuccotto@Nervianoms.com

PMID: 20000735
DOI: 10.1021/jm901443h

No abstract available

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