Lactobionic acid in a natural alkylpolyglucoside-based vehicle: assessing safety and efficacy aspects in comparison to glycolic acid

J Cosmet Dermatol. 2010 Mar;9(1):3-10. doi: 10.1111/j.1473-2165.2010.00474.x.

Abstract

Background/aims: Lactobionic acid (LA) is a newer cosmeceutical active belonging to the class of alpha-hydroxyacids (AHAs), showing advantages over them. The aim of part I of this study was to compare efficacy and irritation potential of LA vs. glycolic acid (GA) from two types of vehicles - gel and emulsion. In part II, effects of LA-containing emulsions based on a new, natural emulsifier of alkylpolyglucoside (APG) type were evaluated.

Methods: Skin bioengineering was used on 77 healthy volunteers to assess: color as erythema and melanin (MI) index, transepidermal water loss, electrical capacitance and pH of the skin. In part I of the study, the parameters were measured after occlusion and periodically during 2 weeks of test samples application; in part II parameters were measured periodically during 4 weeks.

Results/conclusion: LA-containing samples has produced better skin performance when compared with corresponding GA-containing ones, particularly the lack of both skin irritation and skin barrier impairment. When used in vehicles based on a new APG-emulsifier, LA and GA have shown better efficacy, emphasizing the importance of vehicle on the effects of topical actives. LA (6%) in the emulsion based on APGs could be proposed as an alternative to low-molecular AHAs in cosmeceuticals.

Publication types

  • Comparative Study

MeSH terms

  • Administration, Cutaneous
  • Adult
  • Disaccharides / administration & dosage
  • Disaccharides / adverse effects
  • Disaccharides / pharmacology*
  • Emulsions / pharmacology
  • Fatty Alcohols / pharmacology
  • Female
  • Gels / pharmacology
  • Glucosides / pharmacology
  • Glycolates / administration & dosage
  • Glycolates / adverse effects
  • Glycolates / pharmacology*
  • Humans
  • Keratolytic Agents / administration & dosage
  • Keratolytic Agents / adverse effects
  • Keratolytic Agents / pharmacology*
  • Male
  • Pharmaceutical Vehicles / pharmacology
  • Reference Values
  • Skin Irritancy Tests
  • Sunscreening Agents / administration & dosage
  • Sunscreening Agents / adverse effects
  • Sunscreening Agents / pharmacology*

Substances

  • Disaccharides
  • Emulsions
  • Fatty Alcohols
  • Gels
  • Glucosides
  • Glycolates
  • Keratolytic Agents
  • Pharmaceutical Vehicles
  • Sunscreening Agents
  • glycolic acid
  • lactobionic acid