Kinetic studies of chromaffin granule H+-ATPase and effects of bafilomycin A1

Biochem Biophys Res Commun. 1990 Jul 31;170(2):873-8. doi: 10.1016/0006-291x(90)92172-v.

Abstract

Vacuolar type H+-ATPase purified from bovine chromaffin granules did not show simple Michaelis-Menten type kinetics, and had apparent Km values of 5 microM, 30 microM and 300 microM. These three Km values suggested the presence of catalytic cooperativity during steady-state hydrolysis. The single turnover rate was 10(-3)-fold the maximal velocity of the enzyme and similar to the rate estimated from the velocity of steady-state hydrolysis with the smallest Km value (5 microM). The H(+)-ATPase was inhibited by the stoichiometric binding of bafilomycin A1, a specific inhibitor of vacuolar type H(+)-ATPase. This inhibitor not only lowered the rate of ATP hydrolysis at the single catalytic site, but also affected the catalytic cooperativity of the enzyme.

MeSH terms

  • Adenosine Triphosphatases / metabolism*
  • Adenosine Triphosphate / metabolism
  • Animals
  • Anti-Bacterial Agents / pharmacology*
  • Cattle
  • Chromaffin Granules / drug effects
  • Chromaffin Granules / enzymology*
  • Chromaffin System / enzymology*
  • Hydrolysis
  • Kinetics
  • Macrolides*
  • Substrate Specificity

Substances

  • Anti-Bacterial Agents
  • Macrolides
  • bafilomycin A1
  • Adenosine Triphosphate
  • Adenosine Triphosphatases