Control of esophageal distension-induced secondary peristalsis by the GABA(B) agonist baclofen in humans

Neurogastroenterol Motil. 2011 Jul;23(7):612-e250. doi: 10.1111/j.1365-2982.2011.01716.x. Epub 2011 Apr 19.

Abstract

Background: Secondary peristalsis is important for the clearance of retained food bolus or refluxate from the esophagus. The effects of the gamma aminobutyric acid receptor type B (GABA(B) ) agonist on secondary peristalsis remain unclear in humans. We aimed to investigate the effect of a GABA(B) agonist baclofen on esophageal secondary peristalsis.

Methods: After a baseline recording of esophageal motility, secondary peristalsis was generated by slow and rapid mid-esophageal injections of air in 15 healthy subjects. Two separate sessions with 40mg oral baclofen or placebo were randomly performed to test their effects on secondary peristalsis.

Key results: Baclofen increased the threshold volume for triggering secondary peristalsis during slow air distension (P=0.003) and rapid air distension (P=0.002). Baclofen reduced the rate of secondary peristalsis by rapid air distension from 90% to 30% (P=0.0002). Baclofen increased basal lower esophageal sphincter pressure (P=0.03). Baclofen did not affect any of peristaltic parameters during primary or secondary peristalsis.

Conclusions & inferences: This study provides an evidence for inhibitory modulation of esophageal secondary peristalsis by the GABA(B) agonist baclofen. Activation of secondary peristalsis is probably modulated by GABA(B) receptors; however, baclofen does not lead to any motility change in secondary peristalsis.

Publication types

  • Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Adult
  • Baclofen / administration & dosage
  • Baclofen / pharmacology*
  • Dose-Response Relationship, Drug
  • Esophagus / drug effects*
  • Esophagus / physiology
  • Female
  • GABA-B Receptor Agonists / administration & dosage
  • GABA-B Receptor Agonists / pharmacology*
  • Humans
  • Male
  • Manometry
  • Muscle Contraction / drug effects
  • Muscle Contraction / physiology
  • Peristalsis / drug effects*
  • Peristalsis / physiology
  • Receptors, GABA-B / drug effects
  • Receptors, GABA-B / physiology

Substances

  • GABA-B Receptor Agonists
  • Receptors, GABA-B
  • Baclofen