Morphine analgesia and acute physical dependence: rapid onset of two opposing, dose-related processes

Brain Res. 1990 May 14;516(1):37-40. doi: 10.1016/0006-8993(90)90894-h.

Abstract

Enhanced responsiveness to noxious stimulation is a reliable sign of opioid withdrawal and is therefore a measure of physical dependence. In lightly anesthetized rats, naloxone, given i.v. 15 min following i.v. morphine, caused a significant shortening of tail flick latency (hyperalgesia). At each dose of naloxone (0.1, 1.0 or 2.0 mg/kg), the magnitude of the observed hyperalgesia was a function of the preceding dose of morphine (0.5, 1.0 or 2.0 mg/kg). Thus morphine rapidly induces two dose-related opposing processes: one results in antinociception and the other in the potential for hyperalgesia.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Analgesics / pharmacology*
  • Animals
  • Dose-Response Relationship, Drug
  • Male
  • Morphine / pharmacology*
  • Naloxone / pharmacology*
  • Pain / metabolism*
  • Pain / physiopathology
  • Rats
  • Rats, Inbred Strains
  • Receptors, Opioid / drug effects
  • Receptors, Opioid / physiology*
  • Substance Withdrawal Syndrome / physiopathology*
  • Substance-Related Disorders / physiopathology*

Substances

  • Analgesics
  • Receptors, Opioid
  • Naloxone
  • Morphine